SCHEMBL4073906

SCHEMBL4073906

C1CCC2CCCNC2=NC1

nearest known ligand 0.73

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 9/20 0.73
NOS3 P29474 1/20 0.37
NOS1 P29475 1/20 0.37
NOS2 P35228 1/20 0.37
CYP2D6 P10635 2/20 0.33
HTR1A P08908 1/20 0.33
ADRA2A P08913 1/20 0.33
ADRA1A P35348 1/20 0.33
OPRM1 P35372 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
BLM P54132 1/20 0.33
KMT2A Q03164 1/20 0.33
TAAR1 Q96RJ0 1/20 0.33
HRH4 Q9H3N8 1/20 0.32
MAOA P21397 3/20 0.31
MAOB P27338 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10854575 0.96 NISCH (0.73) NISCHNOS3NOS1NOS2CYP2D6
SCHEMBL10852808 0.94 NISCH (0.77) NISCHNOS3NOS1NOS2CYP2D6
SCHEMBL574072 0.93 NISCH (0.69) NISCHNOS3NOS1NOS2CYP2D6
SCHEMBL21391659 0.86 NISCH (0.95) NISCHCYP2D6HTR1AADRA2AADRA1A
SCHEMBL19348515 0.84
SCHEMBL11130232 0.84 NISCH (0.91) NISCHCYP2D6HTR1AADRA2AADRA1A
SCHEMBL1139763 0.84 NISCH (1.00) NISCHCYP2D6HTR1AADRA2AADRA1A
SCHEMBL8142116 0.84 NISCH (1.00) NISCHCYP2D6HTR1AADRA2AADRA1A
SCHEMBL11132739 0.82 NISCH (0.87) NISCHCYP2D6HTR1AADRA2AADRA1A
SCHEMBL11132717 0.80 NISCH (0.83) NISCHCYP2D6HTR1AADRA2AADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090082588-A1 Process for producing fluorinated carbamates and isocyanates REPSOL YPF, S.A. (ES) 2009-03-26 US claimed
EP-2036884-A1 Process for producing fluorinated isocyanates and carbamates REPSOL YPF S.A. (ES) 2009-03-18 EP claimed
CN-107074821-A It is used as the diamines macrocyclic compound of FXIA inhibitor 百时美施贵宝公司 2017-08-18 CN disclosed
US-20090082588-A1 Process for producing fluorinated carbamates and isocyanates REPSOL YPF, S.A. (ES) 2009-03-26 US disclosed
EP-2036884-A1 Process for producing fluorinated isocyanates and carbamates REPSOL YPF S.A. (ES) 2009-03-18 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090082588-A1 Process for producing fluorinated carbamates and isocyanates SRM, CA4, PRMT3 NISCH 27/4885NOS3 167/4885NOS1 244/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.