SCHEMBL4074412

SCHEMBL4074412

c1ccc2c(c1)CCN(C1CCNCC1)CN2

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 8/20 0.43
HTR2B P41595 4/20 0.43
HTR2A P28223 3/20 0.43
TAAR1 Q96RJ0 1/20 0.40
CHRNA7 P36544 1/20 0.40
HRH3 Q9Y5N1 2/20 0.39
HPGD P15428 1/20 0.38
KMT2A Q03164 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
CYP2D6 P10635 1/20 0.37
L3MBTL3 Q96JM7 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6374267 0.84 HTR2C (0.42) HTR2CHTR2BHTR2AHRH3HPGD
SCHEMBL28643716 0.80 HRH3 (0.39) HTR2CHTR2BHTR2AHRH3CYP2D6
SCHEMBL2657988 0.78 SLC18A3 (0.53) HTR2CHTR2BHTR2ATAAR1HRH3
SCHEMBL29501341 0.78 SLC18A3 (0.53) HTR2CHTR2BHTR2ATAAR1HRH3
SCHEMBL2491465 0.77 HRH3 (0.47) HTR2CHTR2BHRH3CYP2D6
Bromide SCHEMBL6423364 0.76 SLC18A3 (0.51) HTR2CHTR2BHTR2ATAAR1HRH3
Hydrochloric Acid SCHEMBL5271851 0.76 SLC18A3 (0.51) HTR2CHTR2BHTR2ATAAR1HRH3
Hydrochloric Acid SCHEMBL29877056 0.76 SLC18A3 (0.51) HTR2CHTR2BHTR2ATAAR1HRH3
Hydrochloric Acid SCHEMBL16835555 0.76 SLC18A3 (0.51) HTR2CHTR2BHTR2ATAAR1HRH3
SCHEMBL28186450 0.75 HRH3 (0.36) HTR2CHTR2BHRH3CYP2D6L3MBTL3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009020470-A2 CGRP RECEPTOR ANTAGONISTS VERTEX PHARMACEUTICALS INCORPORATED (US) 2009-02-12 WO disclosed