SCHEMBL4074526

SCHEMBL4074526

CN(Cc1ncc[nH]1)Cc1nccn1CC(=O)N1CCC2(CCN(C3CCCCC3)CC2)C1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 4/20 0.36
OPRM1 P35372 2/20 0.36
OPRL1 P41146 2/20 0.36
ITGB3 P05106 1/20 0.32
ITGA2B P08514 1/20 0.32
KCNH2 Q12809 1/20 0.32
HRH3 Q9Y5N1 4/20 0.32
CCR4 P51679 1/20 0.31
KMT2A Q03164 1/20 0.31
HSD11B1 P28845 2/20 0.31
PARP1 P09874 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4070832 0.87 CXCR4 (0.39) CXCR4OPRM1OPRL1KCNH2CCR4
SCHEMBL4073706 0.84 CXCR4 (0.51) CXCR4
SCHEMBL4521932 0.82 CXCR4 (0.39) CXCR4
SCHEMBL2695053 0.80 CXCR4 (0.37) CXCR4OPRM1OPRL1ITGB3ITGA2B
SCHEMBL4234443 0.79 HRH3 (0.38) CXCR4ITGB3ITGA2BHRH3
SCHEMBL2694751 0.78 CXCR4 (0.36) CXCR4OPRM1OPRL1ITGB3ITGA2B
SCHEMBL2692227 0.77 HSD11B1 (0.45) CXCR4OPRM1OPRL1KCNH2HRH3
SCHEMBL2694422 0.77 ITGB3 (0.36) CXCR4OPRM1OPRL1ITGB3ITGA2B
SCHEMBL2695480 0.77 CXCR4 (0.36) CXCR4OPRM1OPRL1ITGB3ITGA2B
SCHEMBL2692946 0.77 CXCR4 (0.45) CXCR4HRH3KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2009507867-A 2009-02-26 JP claimed
EP-1928839-A1 METHOD FOR THE PRODUCTION OF 5-FLUORO-1,3-DIALKYL-1H-PYRAZOL-4-CARBONYL FLUORIDES Bayer CropScience AG (DE) 2008-06-11 EP claimed
WO-2007031212-A1 METHOD FOR THE PRODUCTION OF 5-FLUORO-1,3-DIALKYL-1H-PYRAZOL-4-CARBONYL FLUORIDES BAYER CROPSCIENCE AG (DE) 2007-03-22 WO claimed
US-20090325992-A1 COMPOUND HAVING CYCLIC GROUP BOUND THERETO THROUGH SPIRO BINDING AND USE THEREOF ONO PHARMACEUTICAL CO., LTD. (JP) 2009-12-31 US disclosed
EP-2055705-A1 COMPOUND HAVING CYCLIC GROUP BOUND THERETO THROUGH SPIRO BINDING AND USE THEREOF Ono Pharmaceutical CO., LTD. (JP) 2009-05-06 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090325992-A1 COMPOUND HAVING CYCLIC GROUP BOUND THERETO THROUGH SPIRO BINDING AND USE THEREOF CXCR4, CXCL12, CXCR1 CXCR4 1/4885OPRM1 1350/4885OPRL1 397/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.