Dicloralurea

Dicloralurea

SCHEMBL4075855

CN(C)C=O.O=C(NC(O)C(Cl)(Cl)Cl)NC(O)C(Cl)(Cl)Cl

nearest known ligand 0.40

Full drug profile on Sugi Atlas →

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.40
TSHR P16473 1/20 0.36
TDP1 Q9NUW8 1/20 0.32
ALDH1A1 P00352 2/20 0.32
MEN1 O00255 1/20 0.32
MAPT P10636 1/20 0.32
NFKB1 P19838 1/20 0.32
NFKB2 Q00653 1/20 0.32
KMT2A Q03164 1/20 0.32
RELA Q04206 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Dicloralurea SCHEMBL134347 0.82 HPGD (0.45) HPGD
Dicloralurea SCHEMBL6534881 0.78 HPGD (0.41) HPGD
Dicloralurea SCHEMBL2674558 0.76 HPGD (0.41) HPGDALDH1A1MAPT
Dicloralurea SCHEMBL3965395 0.76 HPGD (0.40) HPGDALDH1A1MEN1KMT2A
Dicloralurea SCHEMBL5418303 0.74 HPGD (0.39) HPGDALDH1A1
Mecloralurea SCHEMBL547686 0.74 HPGD (0.44) HPGD
Dicloralurea SCHEMBL17968228 0.73 HPGD (0.41) HPGD
Dicloralurea SCHEMBL4966646 0.71 HPGD (0.39) HPGD
Dicloralurea SCHEMBL6289122 0.71 HPGD (0.36) HPGDALDH1A1
SCHEMBL25292405 0.69 HPGD (0.47) HPGDALDH1A1MEN1MAPTNFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015176025-A9 DISCOIDAL POLYMERIC NANOCONSTRUCTS AND METHODS OF USE IN CANCER THERANOSTICS THE METHODIST HOSPITAL (US) 2015-12-30 WO disclosed
WO-2015176025-A1 DISCOIDAL POLYMERIC NANOCONSTRUCTS AND METHODS OF USE IN CANCER THERANOSTICS THE METHODIST HOSPITAL (US) 2015-11-19 WO disclosed
EP-1188768-B1 LHRH antagonist peptides UNIV INDIANA RES & TECH CORP (US) 2009-06-03 EP disclosed
EP-1725236-A4 NOVEL M3 MUSCARINIC ACETYLCHOLINE RECEPTOR ANTAGONISTS GLAXO GROUP LTD (GB) 2009-05-13 EP disclosed
EP-1751089-A2 NOVEL M3 MUSCARINIC ACETYLCHOLINE RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2007-02-14 EP disclosed
EP-1725236-A1 NOVEL M3 MUSCARINIC ACETYLCHOLINE RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2006-11-29 EP disclosed
US-7071165-B2 LHRH antagonist peptides INDIANA UNIVERSITY RESEARCH AND TECHNOLOGY CORPORATION (US) 2006-07-04 US disclosed
WO-2005087236-A1 NOVEL M3 MUSCARINIC ACETYLCHOLINE RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2005-09-22 WO disclosed
WO-2005086873-A2 NOVEL M3 MUSCARINIC ACETYLCHOLINE RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (US) 2005-09-22 WO disclosed
US-20030181385-A1 LHRH antagonist peptides ADVANCED RESEARCH & TECHNOLOGY INSTITUTE 2003-09-25 US disclosed
US-20030040482-A1 LHRH antagonist peptides ADVANCED RESEARCH & TECHNOLOGY INSTITUTE 2003-02-27 US disclosed
US-6455499-B1 Methods for treating disorders associated with LHRH activity INDIANA UNIVERSITY FOUNDATION 2002-09-24 US disclosed
EP-0794961-B1 LHRH ANTAGONIST PEPTIDES ADVANCED RES & TECH INST (US) 2002-08-28 EP disclosed
US-6423686-B1 LHRH antagonist peptides ADVANCED RESEARCH & TECHNOLOGY INSTITUTE 2002-07-23 US disclosed
EP-1188768-A2 LHRH antagonist peptides Advanced Research & Technology Institute (US) 2002-03-20 EP disclosed
US-5843901-A LHRH antagonist peptides ADVANCED RESEARCH & TECHNOLOGY INSTITUTE (US) 1998-12-01 US disclosed
EP-0794961-A2 LHRH ANTAGONIST PEPTIDES INDIANA UNIVERSITY FOUNDATION (US) 1997-09-17 EP disclosed
WO-1996040757-A2 LHRH ANTAGONIST PEPTIDES INDIANA UNIVERSITY FOUNDATION (US) 1996-12-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030181385-A1 LHRH antagonist peptides LHCGR, GNRHR, PRLHR HPGD 1464/4885TSHR 43/4885TDP1 4856/4885
US-20030040482-A1 LHRH antagonist peptides LHCGR, GNRHR, PRLHR HPGD 1464/4885TSHR 43/4885TDP1 4856/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.