SCHEMBL4075899

SCHEMBL4075899

CCCOc1cc(N)n[nH]1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 4/20 0.41
GAA P10253 3/20 0.41
NPC1 O15118 4/20 0.41
RAB9A P51151 4/20 0.41
TP53 P04637 2/20 0.41
CYP1A2 P05177 2/20 0.41
MAPT P10636 4/20 0.40
GFER P55789 1/20 0.40
KDM4E B2RXH2 3/20 0.37
ALDH1A1 P00352 2/20 0.37
HTT P42858 2/20 0.37
MEN1 O00255 1/20 0.37
USP2 O75604 1/20 0.37
POLB P06746 1/20 0.37
CASP1 P29466 1/20 0.37
CASP7 P55210 1/20 0.37
KMT2A Q03164 1/20 0.37
ATM Q13315 1/20 0.37
TLR8 Q9NR97 1/20 0.36
MCHR1 Q99705 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3020319 0.86
SCHEMBL4275159 0.78 GABRP (0.37) HSD17B10GAANPC1RAB9ATP53
SCHEMBL11008575 0.78 CYP1A2 (0.36) HSD17B10GAANPC1RAB9ATP53
SCHEMBL4017380 0.77 GAA (0.45) HSD17B10GAANPC1RAB9ATP53
SCHEMBL31080659 0.76 GAA (0.40) HSD17B10GAANPC1RAB9ATP53
SCHEMBL9080444 0.75 NPC1 (0.45) HSD17B10GAANPC1RAB9AKDM4E
SCHEMBL161724 0.73
SCHEMBL219145 0.72 ALDH1A1 (0.44) HSD17B10GAATP53MAPTKDM4E
SCHEMBL3338631 0.70 CDK2 (0.38) HSD17B10GAAMCHR1CDK2CDK1
SCHEMBL4069963 0.70 MCHR1 (0.39) HSD17B10GAANPC1RAB9ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1686999-B1 PYRAZOLE DERIVATIVES AS INHIBITORS OF RECEPTOR TYROSINE KINASES ASTRAZENECA AB (SE) 2009-07-01 EP disclosed