Acetic Acid

Acetic Acid

SCHEMBL407645

Brc1ccc(C2CC2)c([Pb])c1.CC(=O)O.CC(=O)O.CC(=O)O

nearest known ligand 0.40

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADRA2AADRA2BADRA2CADRB2AGTR1AVPR1AAVPR1BAVPR2BDKRB2CALCRCHRNA3CHRNB4ESR1ESR2GHSRGNRHRGSC1HSPA8MALT1MC1RMC4RNOS1NOS2NOS3OPRK1OXTRRAMP1RAMP2RAMP3SCN5ASSTR1SSTR2SSTR3SSTR4SSTR5dacAdacBdacCfolPftsImrcAmrcBmrdArplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Acetic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 2/20 0.40
PTGDR Q13258 1/20 0.40
EDNRB P24530 2/20 0.37
EDNRA P25101 2/20 0.37
WDR5 P61964 2/20 0.36
CREBBP Q92793 1/20 0.35
POLB P06746 1/20 0.35
CAMK2A Q9UQM7 1/20 0.35
RARG P13631 2/20 0.34
NOTUM Q6P988 1/20 0.34
RARB P10826 1/20 0.34
ALDH1A1 P00352 1/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
GRK2 P25098 1/20 0.33
CASP6 P55212 1/20 0.33
CASP8 Q14790 1/20 0.33
CTDSP1 Q9GZU7 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acetic Acid SCHEMBL3033132 0.74 MYC (0.40) PTGDR2ALDH1A1MEN1KMT2AKDM4E
SCHEMBL23243079 0.74 KDM4E (0.52) PTGDR2PTGDREDNRBEDNRAWDR5
Acetic Acid SCHEMBL407646 0.72 PTGDR (0.37) PTGDR2PTGDREDNRBEDNRAWDR5
SCHEMBL16957289 0.72 KDM4E (0.36) PTGDR2PTGDRPOLBALDH1A1MEN1
Acetic Acid SCHEMBL3036024 0.72 ALDH1A1 (0.47) POLBALDH1A1KMT2ATDP1KDM4E
Acetic Acid SCHEMBL404308 0.70 PRNP (0.40) PTGDR2POLBALDH1A1MEN1KMT2A
SCHEMBL15567947 0.70 KDM4E (0.47) PTGDR2PTGDRWDR5POLBMEN1
SCHEMBL16905177 0.69 PTGDR (0.40) PTGDR2PTGDRMEN1KMT2AKDM4E
SCHEMBL23243125 0.69 WDR5 (0.45) WDR5POLBALDH1A1MEN1KMT2A
SCHEMBL7401487 0.69 ALDH1A1 (0.53) PTGDR2PTGDRPOLBALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2389066-B1 CYCLOPENTADIONE DERIVED HERBICIDES SYNGENTA LTD (GB) 2017-07-05 EP disclosed
US-8895474-B2 Herbicidally active cyclopentanediones and derivatives thereof, and their use in controlling weeds SYNGENTA LIMITED (GB) 2014-11-25 US disclosed
US-8530388-B2 Cyclopentadione derived herbicides SYNGENTA LIMITED (GB) 2013-09-10 US disclosed
US-20120021912-A1 NOVEL HERBICIDES SYNGENTA CROP PROTECTION LLC (US) 2012-01-26 US disclosed
EP-2389066-A1 CYCLOPENTADIONE DERIVED HERBICIDES Syngenta Limited (GB) 2011-11-30 EP disclosed
EP-2387310-A1 CYCLOPENTADIONE DERIVED HERBICIDES Syngenta Limited (GB) 2011-11-23 EP disclosed
US-20110275515-A1 CYCLOPENTADIONE DERIVED HERBICIDES SYNGENTA CROP PROTECTION, LLC (US) 2011-11-10 US disclosed
US-D646956-S1 TV mount LEUNG ALEX 2011-10-18 US disclosed
WO-2010102848-A1 CYCLOPENTADIONE DERIVED HERBICIDES SYNGENTA LIMITED (GB) 2010-09-16 WO disclosed
WO-2010081894-A1 CYCLOPENTADIONE DERIVED HERBICIDES SYNGENTA LIMITED (GB) 2010-07-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120021912-A1 NOVEL HERBICIDES DDT, CYP4X1, CYP1B1 PTGDR2 2974/4885PTGDR 3226/4885EDNRB 4122/4885
US-20110275515-A1 CYCLOPENTADIONE DERIVED HERBICIDES DDT, CYP1B1, CYP1A1 PTGDR2 1683/4885PTGDR 1469/4885EDNRB 3662/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.