SCHEMBL4079701

SCHEMBL4079701

O=C(CCCC(=O)NCc1cccc(Cl)c1)NCc1cccc(Cl)c1

nearest known ligand 0.65

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.65
GAA P10253 1/20 0.64
NPC1 O15118 1/20 0.59
RAB9A P51151 1/20 0.59
KMT2A Q03164 3/20 0.57
TRPV1 Q8NER1 1/20 0.57
MEN1 O00255 1/20 0.57
TP53 P04637 2/20 0.57
ALDH1A1 P00352 3/20 0.56
TPSAB1 Q15661 1/20 0.56
KDM4E B2RXH2 1/20 0.54
HPGD P15428 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4079697 0.94 SMN1; SMN2 (0.75) SMN1; SMN2GAANPC1RAB9AKMT2A
SCHEMBL11863114 0.92 SMN1; SMN2 (0.57) SMN1; SMN2GAANPC1RAB9AKMT2A
SCHEMBL6646248 0.91 HPGD (0.68) SMN1; SMN2NPC1RAB9AKMT2ATRPV1
SCHEMBL17372428 0.89 KMT2A (0.58) SMN1; SMN2NPC1RAB9AKMT2ATP53
SCHEMBL21183496 0.87 SMN1; SMN2 (0.52) SMN1; SMN2GAANPC1RAB9AKMT2A
SCHEMBL7368316 0.85 TP53 (0.53) SMN1; SMN2NPC1RAB9AKMT2AMEN1
SCHEMBL24499496 0.85 NPC1 (0.61) SMN1; SMN2NPC1RAB9AKMT2AMEN1
SCHEMBL4034877 0.85 ALDH1A1 (0.63) SMN1; SMN2NPC1RAB9AKMT2AMEN1
SCHEMBL1385664 0.85 NPC1 (0.61) SMN1; SMN2NPC1RAB9AKMT2AMEN1
SCHEMBL29625240 0.85 NPC1 (0.61) SMN1; SMN2NPC1RAB9AKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1745010-B1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES GRUENENTHAL GMBH (DE) 2009-08-05 EP claimed
US-20070112007-A1 Cyclohexyl-1, 4-diamine compounds GRUENENTHAL GMBH (DE) 2007-05-17 US claimed
EP-1745010-B1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES GRUENENTHAL GMBH (DE) 2009-08-05 EP disclosed
US-20070112007-A1 Cyclohexyl-1, 4-diamine compounds GRUENENTHAL GMBH (DE) 2007-05-17 US disclosed
EP-1745010-A1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES Grünenthal GmbH (DE) 2007-01-24 EP disclosed
WO-2005110974-A1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES Grünenthal GmbH (DE) 2005-11-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070112007-A1 Cyclohexyl-1, 4-diamine compounds PKD1, DDC, DPYD SMN1; SMN2 1061/4885GAA 20/4885NPC1 46/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.