SCHEMBL4082366

SCHEMBL4082366

c1ccc2c(c1)CC1CCCC[C]21

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.39
CYP19A1 P11511 1/20 0.37
ACHE P22303 1/20 0.36
PTPN1 P18031 2/20 0.36
NOS3 P29474 1/20 0.36
NOS2 P35228 1/20 0.36
CHRNA7 P36544 1/20 0.36
HPGD P15428 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
PTPRC P08575 1/20 0.35
PTPRF P10586 1/20 0.35
CDC25B P30305 1/20 0.35
PLAU P00749 1/20 0.34
CYP2A6 P11509 1/20 0.34
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
SLC18A3 Q16572 1/20 0.34
HTR1A P08908 1/20 0.34
HTR7 P34969 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11297697 0.78 CYP2A6 (0.44) PTPN1NOS3NOS2HPGDL3MBTL1
SCHEMBL8809851 0.76 PLAU (0.46) L3MBTL1PLAUHTR1A
SCHEMBL8555399 0.74 CES1 (0.46) CYP19A1ACHENOS3NOS2L3MBTL1
SCHEMBL16602939 0.69 PDK2 (0.33) PTPN1HPGDL3MBTL1PTPRCPTPRF
SCHEMBL4055026 0.68 MAPT (0.38) TSHRCYP19A1ACHEPTPN1NOS3
SCHEMBL5254581 0.67 ADRA2A (0.49) TSHRHPGDL3MBTL1CYP2A6MAOA
SCHEMBL1022714 0.67 KDM4E (0.45) TSHRCYP19A1PTPN1CHRNA7L3MBTL1
SCHEMBL30436120 0.67 TSHR (0.67) TSHRCYP19A1NOS3NOS2HPGD
SCHEMBL829845 0.64 TSHR (0.48) TSHR
SCHEMBL568779 0.64 TSHR (0.71) TSHRCYP19A1NOS3NOS2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2081600-A1 COMBINATION OF NMDA- RECEPTOR LIGAND AND A COMPOUND WITH 5-HT6 RECEPTOR AFFINITY Laboratorios Del. Dr. Esteve, S.A. (ES) 2009-07-29 EP claimed
WO-2008034815-A1 COMBINATION OF NMDA- RECEPTOR LIGAND AND A COMPOUND WITH 5-HT6 RECEPTOR AFFINITY LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2008-03-27 WO claimed