SCHEMBL4083177

SCHEMBL4083177

CC(NC(=O)CCC(=O)NC1CCC(c2cccs2)(N(C)C)CC1)C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 8/20 0.47
OPRL1 P41146 8/20 0.47
ALDH1A1 P00352 1/20 0.41
RAB9A P51151 4/20 0.40
NPC1 O15118 3/20 0.40
SMN1; SMN2 Q16637 1/20 0.38
TP53 P04637 1/20 0.36
HTT P42858 1/20 0.36
KDM4E B2RXH2 1/20 0.36
KMT2A Q03164 1/20 0.36
CYP3A4 P08684 1/20 0.35
HPGD P15428 1/20 0.35
CYP2C19 P33261 1/20 0.35
SIGMAR1 Q99720 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL206846 0.87 OPRM1 (0.47) OPRM1OPRL1ALDH1A1KMT2ASIGMAR1
SCHEMBL204689 0.84 POLB (0.51) OPRM1OPRL1ALDH1A1HTTKMT2A
SCHEMBL4073137 0.84 OPRM1 (0.43) OPRM1OPRL1ALDH1A1RAB9ANPC1
SCHEMBL4074077 0.84 OPRM1 (0.51) OPRM1OPRL1RAB9ANPC1SMN1; SMN2
SCHEMBL4074080 0.84 OPRM1 (0.51) OPRM1OPRL1RAB9ANPC1SIGMAR1
SCHEMBL4079677 0.81 OPRM1 (0.47) OPRM1OPRL1RAB9ANPC1
SCHEMBL4046091 0.79 ACKR3 (0.50) OPRM1OPRL1ALDH1A1KMT2A
SCHEMBL4081501 0.79 EPHX2 (0.44) OPRM1OPRL1KMT2A
SCHEMBL208376 0.78 OPRM1 (0.44) OPRM1OPRL1ALDH1A1RAB9ANPC1
SCHEMBL206898 0.78 OPRM1 (0.60) OPRM1OPRL1NPC1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1745010-B1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES GRUENENTHAL GMBH (DE) 2009-08-05 EP claimed