SCHEMBL4081501

SCHEMBL4081501

CN(C)C1(c2cccs2)CCC(NC(=O)CCCC(=O)NC(Cc2ccc(Cl)cc2)C(=O)O)CC1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 2/20 0.44
AVPR1A P37288 9/20 0.42
OXTR P30559 1/20 0.41
OPRM1 P35372 2/20 0.41
OPRL1 P41146 2/20 0.41
PTPN2 P17706 1/20 0.40
PTPN1 P18031 1/20 0.40
HDAC1 Q13547 2/20 0.39
HDAC6 Q9UBN7 2/20 0.39
KMT2A Q03164 1/20 0.38
CCKBR P32239 1/20 0.38
CCR2 P41597 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL206439 0.90 HDAC1 (0.42) AVPR1AOXTROPRM1OPRL1HDAC1
SCHEMBL4073137 0.85 OPRM1 (0.43) EPHX2OPRM1OPRL1
SCHEMBL4074077 0.82 OPRM1 (0.51) EPHX2OPRM1OPRL1
SCHEMBL4074080 0.81 OPRM1 (0.51) EPHX2OPRM1OPRL1
SCHEMBL4083177 0.79 OPRM1 (0.47) OPRM1OPRL1KMT2A
SCHEMBL4079677 0.79 OPRM1 (0.47) EPHX2OPRM1OPRL1
SCHEMBL206923 0.78 OPRM1 (0.43) OPRM1OPRL1KMT2A
SCHEMBL4079674 0.76 OPRM1 (0.45) EPHX2OPRM1OPRL1
SCHEMBL4079669 0.76 OPRM1 (0.45) EPHX2OPRM1OPRL1
SCHEMBL4085419 0.76 OPRM1 (0.45) EPHX2OPRM1OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1745010-B1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES GRUENENTHAL GMBH (DE) 2009-08-05 EP claimed