SCHEMBL4083375

SCHEMBL4083375

CC1(C)CN(C2C3CC4CC(O)(C3)CC2(C2CC2)C4)C(=O)N1

nearest known ligand 0.32

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4088855 0.79 HSD11B1 (0.34) HSD11B1
SCHEMBL4089219 0.76 HSD11B1 (0.30) HSD11B1
SCHEMBL76134 0.74 HSD11B1 (0.45) HSD11B1
SCHEMBL4082514 0.69 HSD11B1 (0.37) HSD11B1
SCHEMBL87596 0.68 HSD11B1 (0.42) HSD11B1
SCHEMBL75062 0.68 HSD11B1 (0.42) HSD11B1
SCHEMBL75793 0.68 HSD11B1 (0.42) HSD11B1
SCHEMBL76738 0.67 EPHX2 (0.36) HSD11B1
SCHEMBL4078786 0.66 HSD11B1 (0.34) HSD11B1
SCHEMBL74665 0.64 HSD11B1 (0.44) HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2104665-A2 IMIDAZOLONE AND IMIDAZOLIDINONE DERIVATIVES AS 11B-HSD1 INHIBITORS FOR DIABETES F. Hoffmann-Roche AG (CH) 2009-09-30 EP claimed
WO-2008046758-A2 IMIDAZOLONE AND IMIDAZOLIDINONE DERIVATIVES AS 11B-HSD1 INHIBITORS FOR DIABETES F. HOFFMANN-LA ROCHE AG (CH) 2008-04-24 WO claimed
EP-2104665-A2 IMIDAZOLONE AND IMIDAZOLIDINONE DERIVATIVES AS 11B-HSD1 INHIBITORS FOR DIABETES F. Hoffmann-Roche AG (CH) 2009-09-30 EP disclosed
WO-2008046758-A2 IMIDAZOLONE AND IMIDAZOLIDINONE DERIVATIVES AS 11B-HSD1 INHIBITORS FOR DIABETES F. HOFFMANN-LA ROCHE AG (CH) 2008-04-24 WO disclosed