SCHEMBL4083806

SCHEMBL4083806

Cc1[nH]c(C#Cc2c(-c3ccccc3)noc2C)nc1-c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 5/20 0.45
PTGS2 P35354 5/20 0.45
HPGDS O60760 1/20 0.42
MAPT P10636 2/20 0.40
KMT2A Q03164 3/20 0.40
MEN1 O00255 2/20 0.40
GAA P10253 1/20 0.40
NPSR1 Q6W5P4 1/20 0.39
NPY5R Q15761 1/20 0.39
GABRA5 P31644 3/20 0.38
SMPD3 Q9NY59 1/20 0.38
BRD4 O60885 1/20 0.36
BRD2 P25440 1/20 0.36
CA12 O43570 1/20 0.36
MT-CO2 P00403 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
LMNA P02545 1/20 0.36
CA3 P07451 1/20 0.36
ADRB2 P07550 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3955095 0.77 PTGS1 (0.44) PTGS1PTGS2MAPTKMT2AMEN1
SCHEMBL3951876 0.75 GABRA5 (0.48) PTGS1PTGS2MAPTKMT2AMEN1
SCHEMBL3952892 0.75 PTGS1 (0.44) PTGS1PTGS2MAPTKMT2AMEN1
SCHEMBL3952333 0.74 PTGS1 (0.50) PTGS1PTGS2MAPTKMT2AMEN1
SCHEMBL3958411 0.74 GRM5 (0.53) PTGS1PTGS2KMT2AMEN1GABRA5
SCHEMBL3950844 0.73 PTGS1 (0.45) PTGS1PTGS2MAPTKMT2AMEN1
SCHEMBL3951870 0.72 PTGS1 (0.47) PTGS1PTGS2MAPTKMT2AMEN1
SCHEMBL3951109 0.72 GABRA5 (0.50) PTGS1PTGS2MAPTKMT2AMEN1
SCHEMBL3951121 0.72 PTGS1 (0.44) PTGS1PTGS2MAPTKMT2AMEN1
SCHEMBL6380887 0.71 PTGS2 (0.58) PTGS1PTGS2MAPTKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029559-B1 ARYL-4-ETHYNYL-ISOXAZOLE DERIVATIVES HOFFMANN LA ROCHE (CH) 2009-08-05 EP disclosed