SCHEMBL4084112

SCHEMBL4084112

Cc1ccc(CC2(N(C)C)CCC(NC(=O)CCC(=O)NCCc3ccccc3)CC2)cc1.Cc1cccc(CC2(N(C)C)CCC(NC(=O)CCC(=O)NCCc3ccccc3)CC2)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.45
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
LMNA P02545 2/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
HDAC3 O15379 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC10 Q969S8 1/20 0.42
HDAC11 Q96DB2 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
SSTR1 P30872 1/20 0.42
SSTR4 P31391 1/20 0.42
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
PLAAT3 P53816 1/20 0.41
PLAAT5 Q96KN8 1/20 0.41
PLAAT2 Q9NWW9 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL206736 0.96 HPGD (0.48) HPGDMEN1KMT2ALMNAKDM4E
SCHEMBL208660 0.94 PLAAT3 (0.46) NPC1RAB9APLAAT3PLAAT5PLAAT2
SCHEMBL206578 0.91 ALDH1A1 (0.45) HPGDKMT2ALMNAALDH1A1HDAC3
SCHEMBL207134 0.91 HPGD (0.43) HPGDMEN1KMT2ALMNAKDM4E
SCHEMBL206456 0.91 POLB (0.45) HPGDKMT2ALMNAKDM4EALDH1A1
SCHEMBL207253 0.88 HDAC3 (0.43) HPGDKMT2AALDH1A1HDAC3HDAC1
SCHEMBL207909 0.88 HDAC3 (0.45) HPGDKMT2ALMNAALDH1A1HDAC3
SCHEMBL206288 0.88 ALDH1A1 (0.50) HPGDMEN1KMT2ALMNAALDH1A1
SCHEMBL208454 0.86 ALDH1A1 (0.53) HPGDMEN1KMT2AALDH1A1NPC1
SCHEMBL205912 0.86 HPGD (0.47) HPGDMEN1KMT2ALMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1745010-B1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES GRUENENTHAL GMBH (DE) 2009-08-05 EP claimed