Paraquat

Paraquat

SCHEMBL4084640

C[n+]1ccc(-c2cc[n+](C)cc2)cc1.[Br-].[Br-]

nearest known ligand 0.72

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHKACHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGHRH2OPRM1

The experimentally established mechanism targets of Paraquat. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 2/20 0.72
SLC22A2 O15244 1/20 0.72
SLC22A1 O15245 1/20 0.72
SLC22A3 O75751 1/20 0.72
PABPC1 P11940 1/20 0.62
APOBEC3A P31941 1/20 0.62
EIF4H Q15056 1/20 0.62
APOBEC3G Q9HC16 1/20 0.62
QDPR P09417 2/20 0.58
HDAC8 Q9BY41 3/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Paraquat SCHEMBL21652 0.96 SLC6A4 (0.77) SLC6A4SLC22A2SLC22A1SLC22A3PABPC1
Paraquat SCHEMBL4895671 0.96 SLC6A4 (0.77) SLC6A4SLC22A2SLC22A1SLC22A3PABPC1
Paraquat SCHEMBL22370108 0.93 SLC6A4 (0.72) SLC6A4SLC22A2SLC22A1SLC22A3PABPC1
Paraquat SCHEMBL8331549 0.93 SLC6A4 (0.72) SLC6A4SLC22A2SLC22A1SLC22A3PABPC1
SCHEMBL14596518 0.93 SLC6A4 (0.72) SLC6A4SLC22A2SLC22A1SLC22A3PABPC1
Paraquat SCHEMBL11281521 0.93 SLC6A4 (0.72) SLC6A4SLC22A2SLC22A1SLC22A3PABPC1
Paraquat SCHEMBL21653 0.93 SLC6A4 (0.72) SLC6A4SLC22A2SLC22A1SLC22A3PABPC1
Paraquat SCHEMBL8852265 0.90 SLC22A2 (0.68) SLC6A4SLC22A2SLC22A1SLC22A3PABPC1
Paraquat SCHEMBL30968908 0.90 SLC6A4 (0.68) SLC6A4SLC22A2SLC22A1SLC22A3PABPC1
Paraquat SCHEMBL599615 0.90 SLC22A2 (0.68) SLC6A4SLC22A2SLC22A1SLC22A3PABPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 24 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024132649-A1 HERBICIDAL COMPOSITIONS SYNGENTA CROP PROTECTION AG (CH) 2024-06-27 WO claimed
WO-2020234422-A1 HERBICIDAL COMPOSITIONS SYNGENTA CROP PROTECTION AG (CH) 2020-11-26 WO claimed
US-8337900-B2 Reverse-phase microcapsules for active ingredients, simplified process of manufacture thereof and combined formulation WDG-CS, ZC, EC-SC, and CX FMC CORPORATION 2012-12-25 US claimed
US-20090053271-A1 Reverse-Phase Microcapsules for Actice Ingredients, Simplified Process of Manufacture Thereof and Combined Formulation Wdg- Cs,Zc, Ec-Sc, and Cx FMC CORPORATION 2009-02-26 US claimed
EP-2004718-A1 REVERSE-PHASE MICROCAPSULES FOR ACTIVE INGREDIENTS, SIMPLIFIED PROCESS OF MANUFACTURE THEREOF AND COMBINED FORMULATIONS WDG-CS, ZC, EC-SC AND CX GAT Microencapsulation AG (AT) 2008-12-24 EP claimed
WO-2007112933-A1 REVERSE-PHASE MICROCAPSULES FOR ACTIVE INGREDIENTS, SIMPLIFIED PROCESS OF MANUFACTURE THEREOF AND COMBINED FORMULATIONS WDG-CS, ZC, EC-SC AND CX GAT MICROENCAPSULATION AG (AT) 2007-10-11 WO claimed
JP-54107886-A None JP disclosed
JP-54109086-A None JP disclosed
WO-2024132649-A1 HERBICIDAL COMPOSITIONS SYNGENTA CROP PROTECTION AG (CH) 2024-06-27 WO disclosed
WO-2020234422-A1 HERBICIDAL COMPOSITIONS SYNGENTA CROP PROTECTION AG (CH) 2020-11-26 WO disclosed
US-8337900-B2 Reverse-phase microcapsules for active ingredients, simplified process of manufacture thereof and combined formulation WDG-CS, ZC, EC-SC, and CX FMC CORPORATION 2012-12-25 US disclosed
US-7500895-B2 Patterned substrate, electro-optical device, and method for manufacturing an electro-optical device SEIKO EPSON CORPORATION (JP) 2009-03-10 US disclosed
US-20090053271-A1 Reverse-Phase Microcapsules for Actice Ingredients, Simplified Process of Manufacture Thereof and Combined Formulation Wdg- Cs,Zc, Ec-Sc, and Cx FMC CORPORATION 2009-02-26 US disclosed
US-6455469-B1 SUBSTITUTED ACETANILIDE DERIVATIVE IN COMBINATION WITH OTHER HERBICIDE TO GIVE EFFECTIVE WEED CONTORL ISHIHARA SANGYO KAISHA, LTD. (JP) 2002-09-24 US disclosed
US-4285575-A USING AN ELECTROCHROMIC ELECTROLYTE CONTAINING A CARBOXYLIC-CONTAINING COMPLEXING AGENT, A FERROUS SALT, A METAL SALT, AND A CHROMOGEN; DURABILITY CANON KABUSHIKI KAISHA (JP) 1981-08-25 US disclosed
US-4212518-A ELECTROCHROMIC CELL CANON KABUSHIKI KAISHA (JP) 1980-07-15 US disclosed
JP-S54109086-A IMAGE DISPLAY DEVICE CANON INC 1979-08-27 JP disclosed
JP-S54107886-A IMAGE DISPLAY DEVICE CANON INC 1979-08-24 JP disclosed
US-4153444-A Herbicidal composition KUMIAI CHEMICAL INDUSTRY COMPANY, LTD. (JP) 1979-05-08 US disclosed
US-4028091-A BIPYRIDYLIUM SALTS AND A THIOCARBAMATE KUMIAI CHEMICAL INDUSTRY CO., LTD. (JA) 1977-06-07 US disclosed