SCHEMBL4085419

SCHEMBL4085419

CN(CC(=O)O)C(=O)CCCC(=O)NC1CCC(c2cccs2)(N(C)C)CC1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 9/20 0.45
OPRL1 P41146 9/20 0.45
NPSR1 Q6W5P4 1/20 0.38
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
ALDH1A1 P00352 1/20 0.36
ALOX15 P16050 1/20 0.36
TSHR P16473 1/20 0.36
HSD17B10 Q99714 1/20 0.36
EPHX2 P34913 1/20 0.36
DRD2 P14416 1/20 0.36
DRD4 P21917 1/20 0.36
DRD3 P35462 1/20 0.36
EPHX1 P07099 1/20 0.35
POLB P06746 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4074080 0.91 OPRM1 (0.51) OPRM1OPRL1NPC1RAB9AEPHX2
SCHEMBL4074077 0.89 OPRM1 (0.51) OPRM1OPRL1NPC1RAB9AEPHX2
SCHEMBL208622 0.86 OPRM1 (0.45) OPRM1OPRL1ALDH1A1EPHX2EPHX1
SCHEMBL4079677 0.85 OPRM1 (0.47) OPRM1OPRL1NPC1RAB9AEPHX2
SCHEMBL209213 0.83 OPRM1 (0.41) OPRM1OPRL1NPC1RAB9APOLB
SCHEMBL4079669 0.82 OPRM1 (0.45) OPRM1OPRL1NPC1RAB9AALDH1A1
SCHEMBL4079674 0.82 OPRM1 (0.45) OPRM1OPRL1NPC1RAB9AEPHX2
SCHEMBL251239 0.82 OPRM1 (0.44) OPRM1OPRL1NPC1ALDH1A1TSHR
SCHEMBL251283 0.82 OPRM1 (0.44) OPRM1OPRL1NPC1RAB9AALDH1A1
SCHEMBL4084421 0.82 OPRM1 (0.45) OPRM1OPRL1NPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1745010-B1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES GRUENENTHAL GMBH (DE) 2009-08-05 EP claimed