SCHEMBL4087343

SCHEMBL4087343

CCCNC(=O)N1CC(OC(c2ccccc2Cl)c2ccccc2Cl)C1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 2/20 0.41
MEN1 O00255 1/20 0.41
CYP2C9 P11712 1/20 0.41
KMT2A Q03164 1/20 0.41
FAAH O00519 5/20 0.40
CNR1 P21554 3/20 0.39
CNR2 P34972 3/20 0.39
OPRM1 P35372 3/20 0.39
OPRL1 P41146 3/20 0.39
NAMPT P43490 2/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4075813 0.93 CNR1 (0.46) MEN1KMT2AFAAHCNR1CNR2
SCHEMBL4075586 0.86 NPC1 (0.44) MEN1KMT2AFAAHCNR1CNR2
SCHEMBL5818620 0.85 FAAH (0.50) CYP2C19FAAHCNR1CNR2
SCHEMBL4084883 0.83 HPGD (0.43) MEN1KMT2AFAAHCNR1LMNA
SCHEMBL4077682 0.83 FAAH (0.42) FAAHCNR1CNR2NAMPT
SCHEMBL4075655 0.82 CNR1 (0.51) FAAHCNR1OPRM1OPRL1
SCHEMBL4075572 0.81 CNR1 (0.52) FAAHCNR1CNR2
SCHEMBL4083665 0.81 CNR1 (0.57) FAAHCNR1CNR2
SCHEMBL4083270 0.80 FAAH (0.51) FAAHCNR1CNR2
SCHEMBL4079362 0.80 GAA (0.48) KMT2AFAAHCNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1620395-B1 AZETIDINECARBOXAMIDE DERIVATIVES AND THEIR USE IN THE TREATMENT OF CB1 RECEPTOR MEDIATED DISORDERS VERNALIS RES LTD (GB) 2009-12-30 EP disclosed
US-7504522-B2 Azetidinecarboxamide derivatives and their use in the treatment of cb1 receptor mediated disorders VERNALIS RESEARCH LIMITED (GB) 2009-03-17 US disclosed
US-20070054891-A1 Azetidinecarboxamide derivatives and their use in the treatment of cb1 receptor mediated disorders VERNALIS RESEARCH LIMAITED (GB) 2007-03-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070054891-A1 Azetidinecarboxamide derivatives and their use in the treatment of cb1 receptor mediated disorders CNR1, CNR2, GPR119 CYP2C19 106/4885MEN1 2044/4885CYP2C9 170/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.