SCHEMBL4088596

SCHEMBL4088596

CC(C)C1CC(C(O)COCc2ccc3ccccc3c2)OC1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASR P41180 2/20 0.39
TACR1 P25103 2/20 0.38
MAOB P27338 1/20 0.36
SLC1A3 P43003 1/20 0.34
SLC1A2 P43004 1/20 0.34
SLC1A1 P43005 1/20 0.34
SLC6A2 P23975 3/20 0.34
SLC6A4 P31645 3/20 0.34
SLC6A3 Q01959 3/20 0.34
HTR2A P28223 2/20 0.34
HTR2C P28335 2/20 0.34
HTR2B P41595 2/20 0.34
HTR7 P34969 1/20 0.34
HTR3A P46098 1/20 0.34
HTR4 Q13639 1/20 0.34
CASP1 P29466 1/20 0.34
CASP3 P42574 1/20 0.34
CASP6 P55212 1/20 0.34
CASP8 Q14790 1/20 0.34
ALOX5 P09917 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8171940 1.00 CASR (0.39) CASRTACR1MAOBSLC1A3SLC1A2
SCHEMBL3975545 0.87 HTT (0.44) HTT
SCHEMBL4746758 0.87 HTT (0.44) HTT
SCHEMBL4551129 0.84 TACR1 (0.38) TACR1MAOBHTT
SCHEMBL8178647 0.84 TACR1 (0.38) TACR1MAOBHTT
SCHEMBL4785585 0.81 MAPT (0.37) TACR1SLC1A3SLC1A2SLC1A1
SCHEMBL8172082 0.81 MAPT (0.37) TACR1SLC1A3SLC1A2SLC1A1
SCHEMBL13885022 0.80 TDP1 (0.38) SLC6A4HTT
SCHEMBL4743482 0.80 TACR1 (0.34) TACR1MAOB
SCHEMBL8175955 0.79 TDP1 (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009053277-A1 ASPARTYL PROTEASE INHIBITORS MEDIVIR AB (SE) 2009-04-30 WO disclosed
WO-2008107365-A1 NEW COMPOUNDS MEDIVIR AB (SE) 2008-09-12 WO disclosed