SCHEMBL4092264

SCHEMBL4092264

CCOC(=O)c1c(-c2ccc(OC(F)(F)F)cc2)c2sc(-c3ccc(OC(F)(F)F)cc3)cc2n1Cc1cccc(Cl)c1

nearest known ligand 0.81

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGES O14684 1/20 0.81
TRPV1 Q8NER1 1/20 0.43
PPARG P37231 11/20 0.42
PPARA Q07869 9/20 0.42
TP53 P04637 1/20 0.42
SERPINE1 P05121 1/20 0.41
CYP2C9 P11712 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C19 P33261 1/20 0.41
CYP4X1 Q8N118 1/20 0.41
EGFR P00533 1/20 0.41
CHRM4 P08173 1/20 0.41
ADRB1 P08588 1/20 0.41
ADRA2A P08913 1/20 0.41
ALOX5 P09917 1/20 0.41
ADRB3 P13945 1/20 0.41
DRD2 P14416 1/20 0.41
ADRA2B P18089 1/20 0.41
CHRM3 P20309 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4093589 0.89 PTGES (1.00) PTGESTRPV1PPARGPPARASERPINE1
SCHEMBL4086539 0.88 PTGES (0.62) PTGESTP53SERPINE1KMT2ASMN1; SMN2
SCHEMBL15497056 0.77 PTGES (0.48) PTGESTRPV1PPARGPPARATP53
SCHEMBL4092414 0.75 PTGES (0.72) PTGESSERPINE1CYP2C9CYP1A2CYP2D6
SCHEMBL4086709 0.74 PTGES (0.47) PTGESPPARGTP53KMT2ASMN1; SMN2
SCHEMBL4098784 0.72 TP53 (0.46) PTGESTP53KMT2ASMN1; SMN2MEN1
SCHEMBL4086421 0.71 MAPT (0.48) PTGESTP53KMT2ASMN1; SMN2MEN1
SCHEMBL5812761 0.71 PTGES (0.65) PTGESPPARGPPARASERPINE1PLA2G2A
SCHEMBL15497062 0.71 KMT2A (0.46) PTGESTP53ALOX5KMT2ASMN1; SMN2
SCHEMBL5737792 0.69 PPARG (0.46) PTGESPPARGPPARASERPINE1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090069384-A1 THIENOPYRROLES USEFUL IN THE TREATMENT OF INFLAMMATION BIOLIPOX AB (SE) 2009-03-12 US disclosed
EP-1844051-A1 THIENOPYRROLES USEFUL IN THE TREATMENT OF INFLAMMATION Biolipox AB (SE) 2007-10-17 EP disclosed
WO-2006077412-A1 THIENOPYRROLES USEFUL IN THE TREATMENT OF INFLAMMATION BIOLIPOX AB (SE) 2006-07-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090069384-A1 THIENOPYRROLES USEFUL IN THE TREATMENT OF INFLAMMATION NPY5R, TH, PTGES PTGES 3/4885TRPV1 866/4885PPARG 1385/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.