SCHEMBL40930

SCHEMBL40930

C[C@H]1c2cccc(O)c2C(O)=C2C(=O)[C@]3(O)C(=O)/C(=C(/N)O)C(=O)[C@@H](N(C)C)[C@@H]3[C@@H](O)[C@@H]21

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 10/20 0.73
USP2 O75604 6/20 0.73
HSD17B10 Q99714 6/20 0.73
HIF1A Q16665 3/20 0.73
TSHR P16473 1/20 0.73
KDM4E B2RXH2 9/20 0.72
L3MBTL1 Q9Y468 7/20 0.72
MMP2 P08253 1/20 0.72
MMP3 P08254 1/20 0.72
MMP7 P09237 1/20 0.72
MMP8 P22894 1/20 0.72
ADORA1 P30542 1/20 0.72
ADRA1A P35348 1/20 0.72
MMP13 P45452 1/20 0.72
RECQL P46063 7/20 0.67
PLA2G1B P04054 1/20 0.67
ATG4B Q9Y4P1 1/20 0.67
HPGD P15428 7/20 0.48
MEN1 O00255 6/20 0.48
KMT2A Q03164 6/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23005369 1.00 TDP1 (0.73) TDP1USP2HSD17B10HIF1ATSHR
SCHEMBL21014939 1.00 TDP1 (0.73) TDP1USP2HSD17B10HIF1ATSHR
SCHEMBL4082642 1.00 TDP1 (0.73) TDP1USP2HSD17B10HIF1ATSHR
SCHEMBL4082631 1.00 TDP1 (0.73) TDP1USP2HSD17B10HIF1ATSHR
SCHEMBL1176275 1.00 TDP1 (0.73) TDP1USP2HSD17B10HIF1ATSHR
Water SCHEMBL1649970 0.99 MMP2 (0.74) TDP1USP2HSD17B10HIF1ATSHR
Water SCHEMBL537059 0.97 MMP2 (0.72) TDP1USP2HSD17B10HIF1ATSHR
Alcohol SCHEMBL14973542 0.94 KDM4E (0.72) TDP1USP2HSD17B10HIF1ATSHR
SCHEMBL18610140 0.92 TDP1 (0.65) TDP1USP2HSD17B10HIF1ATSHR
SCHEMBL21793722 0.85 TDP1 (1.00) TDP1USP2HSD17B10HIF1ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 7449 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026060129-A9 FORMULATIONS COMPRISING ENPP1 INHIBITORS Petragen, Inc. (US) 2026-05-21 WO claimed
WO-2026105164-A1 NON-AQUEOUS LIQUID FORMULATIONS OF TETRACYCLINE ANTIBIOTICS ETICO LIFESCIENCES PRIVATE LIMITED (IN) 2026-05-21 WO claimed
US-20260139860-A1 PRODUCTS OF MANUFACTURE FOR THE TREATMENT, PREVENTION AND AMELIORATION OF MICROBIAL INFECTIONS CENTRE FOR DIGESTIVE DISEASES (AU) 2026-05-21 US claimed
EP-3200748-B2 COMPOSITIONS AND METHODS FOR THE TREATMENT AND PROPHYLAXIS OF SURGICAL SITE INFECTIONS POLYPID LTD (IL) 2026-04-15 EP claimed
US-20260091045-A1 PREVENTATIVE MOUTHWASH CONTAINING DOXYCYCLINE AND METHOD OF PREVENTING COVID INFECTION USING THE PREVENTATIVE MOUTHWASH ROSEMAN BRUCE (US) 2026-04-02 US claimed
US-20260053823-A1 PREVENTATIVE MOUTHWASH CONTAINING A SUB-ANTIMICROBIAL ORAL DOSAGE OF DOXYCYCLINE, METHOD OF PREVENTING COVID INFECTION USING THE MOUTHWASH, AND METHOD OF FORMULATING THE MOUTHWASH ROSEMAN BRUCE (US) 2026-02-26 US claimed
US-20260041701-A1 PHARMACEUTICAL COMPOSITIONS AND METHODS OF MAKING ON DEMAND SOLID DOSAGE FORMULATIONS EASTERN VIRGINIA MEDICAL SCHOOL (US) 2026-02-12 US claimed
EP-4680248-A1 PRODUCTS OF MANUFACTURE AND THERAPEUTIC COMPOSITIONS FOR TREATING, AMELIORATING OR PREVENTING VIRAL INFECTIONS AND METHODS FOR MAKING AND USING THEM Topelia Aust Limited (ACN 652 771 670) (AU) 2026-01-21 EP claimed
EP-4662203-A1 BINDARIT CONJUGATES, COMPOSITIONS AND METHODS FOR TREATING OCULAR DISEASES OR DISORDERS Translatum Medicus Inc. (CA) 2025-12-17 EP claimed
US-20250269005-A1 METHODS FOR TREATING, AMELIORATING OR PREVENTING INFECTIONS USING DRUG AND VACCINATION COMBINATION TREATMENT TOPELIA AUST LIMITED (ACN 652 771 670) (AU) 2025-08-28 US claimed
EP-0374531-B1 Method for the treatment of periodontal disease by sustained delivery of a therapeutic agent to the periodontal pocket, composition of matter therefor and apparatus for the administration thereof AMERICAN CYANAMID CO (US) 1994-05-04 EP claimed
WO-1993024154-A1 BIODEGRADABLE CONTROLLED RELEASE MELT-SPUN DELIVERY SYSTEM FUISZ TECHNOLOGIES, LTD. (US) 1993-12-09 WO claimed
US-5188836-A SUSTAINED RELEASE FORMULATIONS WARNER-LAMBERT COMPANY (US) 1993-02-23 US claimed
US-5167964-A Coating of blend of ethyl acrylate-methacrylic acid copolymer and povidone WARNER-LAMBERT COMPANY (US) 1992-12-01 US claimed
US-5122519-A Tetracyclines in solvent, gelling vehicle AMERICAN CYANAMID COMPANY (US) 1992-06-16 US claimed
WO-1992004902-A1 BIODEGRADABLE GEL MICRO VESICULAR SYSTEMS, INC. (US) 1992-04-02 WO claimed
EP-0470047-A1 Sustained release formulations WARNER-LAMBERT COMPANY (US) 1992-02-05 EP claimed
EP-0374531-A2 Method for the treatment of periodontal disease by sustained delivery of a therapeutic agent to the periodontal pocket, composition of matter therefor and apparatus for the administration thereof AMERICAN CYANAMID COMPANY (US) 1990-06-27 EP claimed
EP-0337733-A2 Single dose intramuscular treatment of chlamydia trachomatis infections PFIZER INC. (US) 1989-10-18 EP claimed
US-4678512-A Marine coating compositions and method GRAMS RALPH R 1987-07-07 US claimed