SCHEMBL41022

SCHEMBL41022

COc1ccc(C(c2ccc(OC)cc2)c2ccc(OC)cc2)cc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 1/20 0.71
CA1 P00915 2/20 0.65
CA2 P00918 2/20 0.65
CA7 P43166 2/20 0.65
CA9 Q16790 2/20 0.65
CA12 O43570 1/20 0.65
CA14 Q9ULX7 1/20 0.65
TDP1 Q9NUW8 4/20 0.56
MAPK1 P28482 3/20 0.56
ALDH1A1 P00352 2/20 0.56
L3MBTL1 Q9Y468 2/20 0.56
TSHR P16473 1/20 0.56
ACHE P22303 1/20 0.52
CYP1A2 P05177 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C19 P33261 1/20 0.50
KDM4E B2RXH2 1/20 0.48
NPC1 O15118 1/20 0.48
GAA P10253 1/20 0.48
MAPT P10636 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16859725 1.00 SLC2A1 (0.71) SLC2A1CA1CA2CA7CA9
SCHEMBL13317344 0.90 ACHE (0.71) SLC2A1CA1CA2CA7CA9
SCHEMBL6347435 0.90 ACHE (0.71) SLC2A1CA1CA2CA7CA9
SCHEMBL34971 0.90 SLC2A1 (0.61) SLC2A1CA1CA2CA7CA9
SCHEMBL40557 0.90 SLC2A1 (0.61) SLC2A1CA1CA2CA7CA9
SCHEMBL14205685 0.90 SLC2A1 (0.61) SLC2A1CA1CA2CA7CA9
SCHEMBL16865571 0.90 ACHE (0.71) SLC2A1CA1CA2CA7CA9
SCHEMBL13295540 0.90 SLC2A1 (0.61) SLC2A1CA1CA2CA7CA9
SCHEMBL13295537 0.90 SLC2A1 (0.61) SLC2A1CA1CA2CA7CA9
SCHEMBL13295535 0.90 SLC2A1 (0.61) SLC2A1CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 4953 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2991655-B1 COMPOSITIONS AND METHODS FOR ALTERING SECOND MESSENGER SIGNALING MEMORIAL SLOAN KETTERING CANCER CENTER (US) 2024-04-10 EP claimed
WO-2024044792-A1 UNIVERSAL SOLID SUPPORTS AND PHOSPHORAMIDITE BUILDING BLOCKS FOR OLIGONUCLEOTIDE SYNTHESIS AM CHEMICALS LLC (US) 2024-02-29 WO claimed
EP-3643706-B1 MODIFIED NUCLEIC ACID MONOMERS AND OLIGONUCLEIC ACID ANALOGUES, WITH HIGH BIOLOGICAL STABILITY AND TARGET GENE SILENCING ACTIVITY, FOR USE IN THERAPY AND DIAGNOSIS OF CANCER AND VIRAL DISEASES EISAI R&D MAN CO LTD (JP) 2023-11-15 EP claimed
EP-3606528-B1 TRICYCLIC COMPOUNDS AS GLYCOGEN SYNTHASE KINASE 3 (GSK3) INHIBITORS AND USES THEREOF BROAD INST INC (US) 2023-10-18 EP claimed
EP-3649135-B1 SYNTHESIS OF HALICHONDRINS HARVARD COLLEGE (US) 2022-12-28 EP claimed
US-11241435-B2 Uses of salt-inducible kinase (SIK) inhibitors for treating osteoporosis THE GENERAL HOSPITAL CORPORATION (US) 2022-02-08 US claimed
EP-3898841-A1 ASYMMETRIC RHODAMINE DYE AND USE THEREOF IN BIOLOGICAL ASSAYS Life Technologies Corporation (US) 2021-10-27 EP claimed
EP-3898842-A1 MODIFIED RHODAMINE DYE AND USE THEREOF IN BIOLOGICAL ASSAYS Life Technologies Corporation (US) 2021-10-27 EP claimed
EP-3172213-B1 MACROCYCLIC KINASE INHIBITORS AND USES THEREOF DANA FARBER CANCER INST INC (US) 2021-09-22 EP claimed
EP-3092220-B1 VITAMIN C PRODRUGS AND USES THEREOF UNIV FLORIDA (US) 2021-01-20 EP claimed
US-4725677-A USING PHOSPHINE DERIVATIVE BIOSYNTECH GMBH (DE) 1988-02-16 US claimed
US-4631339-A 1,3,5-triazepinones ELI LILLY AND COMPANY (US) 1986-12-23 US claimed
US-4461906-A IMPROVING INTELLECTUAL CAPACITY HOFFMANN-LA ROCHE INC. (US) 1984-07-24 US claimed
US-4452807-A CENTRAL NERVOUS SYSTEM DISORDERS HOFFMANN-LA ROCHE INC. (US) 1984-06-05 US claimed
US-4407750-A Unsymmetrical azetidinone aldehyde disulfides and process ELI LILLY AND COMPANY (US) 1983-10-04 US claimed
US-4394313-A Symmetrical azetidinone aldehyde disulfides and process ELI LILLY AND COMPANY (US) 1983-07-19 US claimed
US-4335240-A Process for cyclization ELI LILLY AND COMPANY (US) 1982-06-15 US claimed
US-4302391-A Unsymmetrical azetidinone aldehyde disulfides and process ELI LILLY AND COMPANY (US) 1981-11-24 US claimed
US-4293495-A Symmetrical azetidinone aldehyde disulfides and process ELI LILLY AND COMPANY (US) 1981-10-06 US claimed
US-4293493-A Azetidinone alcohol disulfides and process for cyclization ELI LILLY AND COMPANY (US) 1981-10-06 US claimed