SCHEMBL410243

SCHEMBL410243

O=C1CCC(N2C(=O)c3ccccc3C2=O)C(=O)O1

nearest known ligand 0.55

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 17/20 0.55
DDB1 Q16531 15/20 0.55
IKZF3 Q9UKT9 2/20 0.55
ALDH1A1 P00352 1/20 0.55
CHRM2 P08172 1/20 0.55
OPRM1 P35372 1/20 0.55
CYP1A2 P05177 1/20 0.55
TSHR P16473 1/20 0.55
TDP1 Q9NUW8 1/20 0.55
TNF P01375 1/20 0.43
IL1B P01584 1/20 0.43
TBXA2R P21731 1/20 0.43
IKZF1 Q13422 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL410700 1.00 CRBN (0.55) CRBNDDB1IKZF3ALDH1A1CHRM2
SCHEMBL7284377 1.00 CRBN (0.55) CRBNDDB1IKZF3ALDH1A1CHRM2
SCHEMBL442296 1.00 CRBN (0.55) CRBNDDB1IKZF3ALDH1A1CHRM2
SCHEMBL20075961 0.84 GAA (0.46) CRBNDDB1IKZF3ALDH1A1CHRM2
SCHEMBL10074225 0.84 DDB1 (0.61) CRBNDDB1IKZF3ALDH1A1CHRM2
SCHEMBL11606116 0.83 DDB1 (0.46) CRBNDDB1IKZF3ALDH1A1CHRM2
SCHEMBL986701 0.83 DDB1 (0.46) CRBNDDB1IKZF3ALDH1A1CHRM2
SCHEMBL14601082 0.80 DDB1 (0.44) CRBNDDB1IKZF3ALDH1A1CHRM2
SCHEMBL14377303 0.79 DDB1 (0.65) CRBNDDB1IKZF3ALDH1A1CYP1A2
SCHEMBL15930060 0.79 DDB1 (0.65) CRBNDDB1IKZF3ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 260 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116769191-A Preparation of amygdalin and application of amygdalin in health care products for enhancing immunity 杨振东 2023-09-19 CN claimed
CN-110643670-A Method for preparing D-glutamine by chemical enzyme method 湖北新生源生物工程有限公司 2020-01-03 CN claimed
JP-55036453-A None JP disclosed
EP-4730479-A2 FLAME-RETARDANT NON-AQUEOUS ELECTROLYTIC SOLUTION AND SECONDARY BATTERY USING SAME Kyoto University (JP) 2026-04-22 EP disclosed
EP-4127157-B1 MODIFIED DIPEPTIDE CLEAVASES, USES THEREOF AND RELATED KITS ENCODIA INC (US) 2026-02-11 EP disclosed
EP-4649963-A2 IMIDE-BASED MODULATORS OF PROTEOLYSIS AND ASSOCIATED METHODS OF USE Arvinas Operations, Inc. (US) 2025-11-19 EP disclosed
EP-3131588-B1 IMIDE-BASED MODULATORS OF PROTEOLYSIS AND ASSOCIATED METHODS OF USE ARVINAS OPERATIONS INC (US) 2025-11-05 EP disclosed
US-20250246685-A1 FLAME-RETARDANT NON-AQUEOUS ELECTROLYTIC SOLUTION AND SECONDARY BATTERY USING SAME KYOTO UNIVERSITY (JP) 2025-07-31 US disclosed
WO-2025120994-A1 SECONDARY BATTERY NON-AQUEOUS ELECTROLYTE AND SECONDARY BATTERY PROVIDED WITH SAME ステラケミファ株式会社 2025-06-12 WO disclosed
WO-2025095088-A1 NON-AQUEOUS ELECTROLYTE SOLUTION FOR SECONDARY BATTERY, AND SECONDARY BATTERY PROVIDED WITH SAID SOLUTION ステラケミファ株式会社 2025-05-08 WO disclosed
EP-4509184-A2 COMPOUNDS AND METHODS FOR THE TARGETED DEGRADATION OF ANDROGEN RECEPTOR Arvinas Operations, Inc. (US) 2025-02-19 EP disclosed
WO-2001041755-A2 TOPICAL COMPOSITIONS COMPRISING THALIDOMIDE FOR THE TREATMENT OF INFLAMMATORY DISEASES THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2001-06-14 WO disclosed
EP-1091726-A2 ANALOGS OF 2-PHTHALIMIDINOGLUTARIC ACID AND THEIR USE AS INHIBITORS OF ANGIOGENESIS EntreMed, Inc. (US) 2001-04-18 EP disclosed
US-6161544-A Methods for accelerated orthokeratology KERATOFORM, INC. (US) 2000-12-19 US disclosed
EP-1051655-A1 METHODS AND APPARATUS FOR ACCELERATED ORTHOKERATOLOGY Ista Pharmaceuticals, Inc. (US) 2000-11-15 EP disclosed
WO-1999058096-A9 ANALOGS OF 2-PHTHALIMIDINOGLUTARIC ACID AND THEIR USE AS INHIBITORS OF ANGIOGENESIS ENTREMED INC (US) 2000-07-13 WO disclosed
WO-1999058096-A2 ANALOGS OF 2-PHTHALIMIDINOGLUTARIC ACID AND THEIR USE AS INHIBITORS OF ANGIOGENESIS ENTREMED, INC. (US) 1999-11-18 WO disclosed
WO-1999039238-A1 METHODS AND APPARATUS FOR ACCELERATED ORTHOKERATOLOGY KERATOFORM, INC. (US) 1999-08-05 WO disclosed
JP-S5536453-A NOVEL IMMUNOSUPPRESSIVE AGENT MITSUBISHI CHEM IND LTD 1980-03-14 JP disclosed
US-4087331-A CATALYTICALLY REACTING THE ENZYME WITH A SYNTHETIC PEPTIDE OF GLUTAMIC ACID, DIAZOTIZING THE CLEAVAGE PRODUCT COULTER ELECTRONICS, INC. (US) 1978-05-02 US disclosed