SCHEMBL41100

SCHEMBL41100

CC(=O)OC(C)OC(=O)C1=C(COC(N)=O)CSC2C(NC(=O)/C=N/OCc3ccco3)C(=O)N12

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCC4 O15439 1/20 0.67
PDE4A P27815 1/20 0.67
TDP1 Q9NUW8 8/20 0.50
HSD17B10 Q99714 6/20 0.50
NR1I2 O75469 2/20 0.50
PGR P06401 1/20 0.50
ALDH1A1 P00352 1/20 0.50
TSHR P16473 1/20 0.50
MAPT P10636 8/20 0.49
CTDSP1 Q9GZU7 3/20 0.49
POLB P06746 2/20 0.49
PKM P14618 2/20 0.49
MAPK1 P28482 2/20 0.49
PTGS1 P23219 2/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
HPGD P15428 2/20 0.42
DNMT1 P26358 1/20 0.42
SLC22A6 Q4U2R8 1/20 0.42
SLC22A8 Q8TCC7 1/20 0.42
SLC22A11 Q9NSA0 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6651040 0.87 TDP1 (0.62) ABCC4PDE4ATDP1HSD17B10NR1I2
SCHEMBL10764999 0.87 TDP1 (0.62) ABCC4PDE4ATDP1HSD17B10NR1I2
SCHEMBL11238964 0.84 TDP1 (0.60) TDP1HSD17B10NR1I2PGRALDH1A1
Cefuroxime Axetil SCHEMBL721709 0.80 ABCC4 (1.00) ABCC4PDE4ATDP1HSD17B10NR1I2
Cefuroxime Axetil SCHEMBL10556419 0.80 ABCC4 (1.00) ABCC4PDE4ATDP1HSD17B10NR1I2
Cefuroxime Axetil SCHEMBL379336 0.80 ABCC4 (1.00) ABCC4PDE4ATDP1HSD17B10NR1I2
Cefuroxime Axetil SCHEMBL13575811 0.80 ABCC4 (1.00) ABCC4PDE4ATDP1HSD17B10NR1I2
Cefuroxime Axetil SCHEMBL7767287 0.80 ABCC4 (1.00) ABCC4PDE4ATDP1HSD17B10NR1I2
Cefuroxime Axetil SCHEMBL41099 0.80 ABCC4 (1.00) ABCC4PDE4ATDP1HSD17B10NR1I2
Cefuroxime Axetil SCHEMBL6859269 0.80 ABCC4 (1.00) ABCC4PDE4ATDP1HSD17B10NR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 8879 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4740962-A1 PHARMACEUTICAL COMPOSITION, FORMULATION CONTAINING PHARMACEUTICAL COMPOSITION, KIT CONTAINING PHARMACEUTICAL COMPOSITION, PREPARATION METHOD FOR PHARMACEUTICAL COMPOSITION, AND USE OF PHARMACEUTICAL COMPOSITION Shanghai WD Pharmaceutical Co., Ltd (CN) 2026-05-13 EP claimed
US-20260098299-A1 GENE EXPRESSION-BASED IDENTIFICATION OF EARLY LYME DISEASE THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2026-04-09 US claimed
US-20260048013-A1 PHARMACEUTICAL FORMULATION WITH IMPROVED SOLUBILITY AND BIOAVAILABILITY CONSEJO SUPERIOR INVESTIGACION (ES) 2026-02-19 US claimed
EP-4071477-B1 COMPOSITIONS AND METHODS FOR DIAGNOSING LYME DISEASE AND FOR PREDICTING LYME DISEASE SPIROCHETE ELIMINATION AFTER TREATMENT QIAGEN SCIENCES LLC (US) 2026-01-21 EP claimed
EP-3452124-B1 HEMOSTATIC DEVICES AND METHODS OF USE MEDTRONIC INC (US) 2025-10-08 EP claimed
EP-3452123-B1 HEMOSTATIC DEVICES AND METHODS OF USE MEDTRONIC INC (US) 2025-09-24 EP claimed
US-20250271428-A1 PEPTIDE-BASED BIOMARKERS AND RELATED ASPECTS FOR DISEASE DETECTION ARIZONA BOARD OF REGENTS ON BEHALF OF ARIZONA STATE UNIVERSITY (US) 2025-08-28 US claimed
US-20250222118-A1 Beta-Lactam-Cannabinoid Conjugate Molecules DIVERSE BIOTECH INC (US) 2025-07-10 US claimed
EP-3230500-B1 METHODS OF ORIENTING MULTIFILAMENT YARN AND MONOFILAMENTS OF POLY-4-HYDROXYBUTYRATE AND COPOLYMERS THEREOF TEPHA INC (US) 2025-06-18 EP claimed
EP-4566590-A1 TASTE-MASKING MICROSPHERE, PREPARATION PROCESS THEREFOR, AND USE THEREOF Harbin Kanon Pharmaceutical Co., Ltd (CN) 2025-06-11 EP claimed
EP-0422290-A1 Novel drug delivery system ELI LILLY AND COMPANY (US) 1991-04-17 EP claimed
EP-0223365-B1 CEFUROXIME AXETIL DRAGEE GLAXO GROUP LIMITED (GB) 1991-02-27 EP claimed
US-4994567-A Purification by recovering from solution by roller drying GALAXO GROUP LIMITED (GB) 1991-02-19 US claimed
US-4897270-A Coated tablet containing cefuroxime axetil GLAXO GROUP LIMITED 1990-01-30 US claimed
US-4865851-A WITH WATER INSOLUBLE LIPID COATING TO MASK BITTER TASTE GLAXO GROUP LIMITED (GB) 1989-09-12 US claimed
US-4820833-A PURIFICATION BY SPRAY DRYING PRECIPITATION, FREEZE DRYING; CEPHALOSPORINS GLAXO GROUP LIMITED (GB) 1989-04-11 US claimed
CN-88102851-A METHOD FOR PREPARING PHARMACEUTICAL COMPOSITION 1988-12-21 CN claimed
EP-0223365-A2 Cefuroxime axetil dragee GLAXO GROUP LIMITED (GB) 1987-05-27 EP claimed
US-4562181-A INCREASED ABSORPTION VIA THE GASTROINTESTINAL TRACT, ALLOWING FOR ORAL OR RECTAL ADMINISTRATION GLAXO GROUP LIMITED (GB) 1985-12-31 US claimed
EP-0107276-A2 Novel form of cefuroxime ester, process for its preparation and composition containing it GLAXO GROUP LIMITED (GB) 1984-05-02 EP claimed