SCHEMBL4115545

SCHEMBL4115545

O=[N+]([O-])c1cnc(Cl)nc1Nc1ccc2[nH]ncc2c1

nearest known ligand 0.64

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HSF1 Q00613 1/20 0.64
PIN1 Q13526 1/20 0.60
MKNK1 Q9BUB5 3/20 0.50
POLB P06746 1/20 0.48
MAPT P10636 1/20 0.48
MAOB P27338 1/20 0.48
NOS1 P29475 1/20 0.48
ROCK2 O75116 7/20 0.46
ROCK1 Q13464 3/20 0.46
KDR P35968 2/20 0.45
EGFR P00533 1/20 0.45
MAPKAPK2 P49137 1/20 0.44
GSK3B P49841 1/20 0.43
SYK P43405 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23931958 0.91 PIN1 (0.60) HSF1PIN1MAPTNOS1KDR
SCHEMBL6789738 0.85 HSF1 (0.72) HSF1MKNK1POLBMAPTMAOB
SCHEMBL12612614 0.82 PIN1 (0.58) HSF1PIN1POLBMAPTMAOB
SCHEMBL16638034 0.81 ROCK2 (0.64) MKNK1ROCK2ROCK1KDREGFR
SCHEMBL6787283 0.80 HSF1 (0.72) HSF1MKNK1POLBMAPTMAOB
SCHEMBL29695654 0.80 HSF1 (0.65) HSF1MKNK1POLBMAPTMAOB
SCHEMBL657293 0.79 ROCK2 (0.61) MKNK1ROCK2ROCK1SYK
SCHEMBL2442475 0.79 MKNK1 (0.59) MKNK1MAPTROCK2ROCK1KDR
SCHEMBL15639737 0.79 MKNK1 (0.55) MKNK1ROCK2ROCK1KDREGFR
SCHEMBL29974061 0.79 PIN1 (0.79) PIN1POLBMAPTGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009063240-A1 2,4-DIAMINOPYRIMIDINE DERIVATIVES USEFUL AS INHIBITORS OF AURORA KINASE ARROW THERAPEUTICS LIMITED (GB) 2009-05-22 WO disclosed