SCHEMBL4124009

SCHEMBL4124009

Fc1ccc(-c2cc([AsH]c3ccc(OC(F)(F)F)cc3)cc(N3CCOCC3)n2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 2/20 0.47
AKT1 P31749 1/20 0.47
MTOR P42345 1/20 0.47
PRKDC P78527 2/20 0.46
ABL1 P00519 4/20 0.44
BCR P11274 1/20 0.44
RAB9A P51151 2/20 0.44
NPC1 O15118 1/20 0.44
AR P10275 1/20 0.44
TSHR P16473 4/20 0.43
NPSR1 Q6W5P4 3/20 0.43
KDM4E B2RXH2 2/20 0.43
HPGD P15428 2/20 0.43
HSD17B10 Q99714 2/20 0.43
ALDH1A1 P00352 1/20 0.43
KMT2A Q03164 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
SCN9A Q15858 2/20 0.41
MAPT P10636 1/20 0.40
MAPK1 P28482 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5195190 0.84 NPSR1 (0.46) PIK3CAAKT1MTORPRKDCABL1
SCHEMBL4358342 0.82 ABL1 (0.56) PIK3CAAKT1MTORPRKDCABL1
SCHEMBL28042881 0.78 ABL1 (0.49) PIK3CAAKT1MTORPRKDCABL1
SCHEMBL28043071 0.78 ABL1 (0.52) PIK3CAAKT1MTORPRKDCABL1
SCHEMBL3999646 0.74 L3MBTL1 (0.55) ABL1NPSR1KDM4EHPGDALDH1A1
SCHEMBL3451786 0.73 ABL1 (0.63) PIK3CAAKT1MTORABL1BCR
SCHEMBL3232353 0.71 TSHR (0.56) PIK3CAPRKDCRAB9ANPC1AR
SCHEMBL3450413 0.70 ABL1 (0.56) PIK3CAAKT1MTORABL1BCR
SCHEMBL3997867 0.70 L3MBTL1 (0.50) ABL1BCRKDM4EKMT2A
SCHEMBL4002840 0.69 SCN9A (0.46) ABL1BCRKDM4EALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1805142-A4 NOVEL PYRIDINE COMPOUNDS, PROCESS FOR THEIR PREPARATION AND COMPOSITIONS CONTAINING THEM REDDY US THERAPEUTICS INC (US) 2009-06-10 EP disclosed
EP-1805142-A2 NOVEL PYRIDINE COMPOUNDS, PROCESS FOR THEIR PREPARATION AND COMPOSITIONS CONTAINING THEM Reddy US Therapeutics, Inc. (US) 2007-07-11 EP disclosed
WO-2006034474-A2 NOVEL PYRIDINE COMPOUNDS, PROCESS FOR THEIR PREPARATION AND COMPOSITIONS CONTAINING THEM REDDY US THERAPEUTICS, INC. (US) 2006-03-30 WO disclosed