SCHEMBL28043071

SCHEMBL28043071

CNc1cc(-c2ccc(OC(F)(F)F)cc2)nc(N2CCOCC2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 5/20 0.52
BCR P11274 2/20 0.52
PRKDC P78527 1/20 0.48
KDM4E B2RXH2 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
AKT1 P31749 2/20 0.47
PIK3CA P42336 1/20 0.47
MTOR P42345 1/20 0.47
MCHR1 Q99705 1/20 0.47
GRM2 Q14416 2/20 0.44
CTSS P25774 1/20 0.44
CTSK P43235 1/20 0.44
RAF1 P04049 1/20 0.43
BRAF P15056 1/20 0.43
NPSR1 Q6W5P4 2/20 0.43
MAPT P10636 1/20 0.43
TSHR P16473 1/20 0.43
MAPK1 P28482 1/20 0.43
HSD17B10 Q99714 1/20 0.43
SCN9A Q15858 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28042885 0.90 GALR2 (0.51) ABL1BCRKDM4EMCHR1MAPT
SCHEMBL4358342 0.85 ABL1 (0.56) ABL1BCRPRKDCKDM4ETDP1
SCHEMBL28043075 0.85 NPSR1 (0.47) KDM4ETDP1AKT1PIK3CAMTOR
SCHEMBL28042881 0.80 ABL1 (0.49) ABL1BCRPRKDCKDM4ETDP1
SCHEMBL4124009 0.78 PIK3CA (0.47) ABL1BCRPRKDCKDM4ETDP1
SCHEMBL4358479 0.77 ABL1 (0.55) ABL1BCRKDM4EAKT1PIK3CA
SCHEMBL3450413 0.77 ABL1 (0.56) ABL1BCRTDP1AKT1PIK3CA
SCHEMBL3996650 0.76 ABL1 (0.56) ABL1BCRAKT1PIK3CAMTOR
SCHEMBL3997867 0.74 L3MBTL1 (0.50) ABL1BCRKDM4EMCHR1PIM1
SCHEMBL4281796 0.74 ABL1 (0.48) ABL1BCRAKT1PIK3CAMTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105143188-A Novel sulfonamide trpa1 receptor antagonists PHARMESTE S R L IN LIQUIDATION 2015-12-09 CN disclosed