SCHEMBL4128827

SCHEMBL4128827

CCOC(=O)CN1CCC(CN(CC2CCCCC2)c2nc3c(C(C)(C)C)nn(C)c3c(=O)[nH]2)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 3/20 0.37
NPSR1 Q6W5P4 2/20 0.36
MAPT P10636 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
POLB P06746 2/20 0.35
LMNA P02545 2/20 0.34
HTT P42858 1/20 0.34
HIF1A Q16665 1/20 0.34
MCOLN3 Q8TDD5 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.33
NPY1R P25929 1/20 0.33
GAA P10253 1/20 0.33
MAPK1 P28482 1/20 0.33
PDE5A O76074 4/20 0.32
ABCC5 O15440 1/20 0.32
GSK3B P49841 1/20 0.32
PDE1A P54750 1/20 0.31
PDE1B Q01064 1/20 0.31
PDE1C Q14123 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4127434 0.89 KDM4E (0.35) KDM4EALDH1A1NPSR1MAPTSMN1; SMN2
SCHEMBL8045132 0.85 KDM4E (0.41) KDM4EALDH1A1NPSR1MAPTSMN1; SMN2
SCHEMBL4122386 0.83 KDM4E (0.36) KDM4EALDH1A1NPSR1MAPTSMN1; SMN2
SCHEMBL4140662 0.83 KDM4E (0.35) KDM4EALDH1A1NPSR1MAPTSMN1; SMN2
SCHEMBL4139405 0.82 KDM4E (0.34) KDM4EALDH1A1NPSR1MAPTSMN1; SMN2
SCHEMBL8043827 0.82 KDM4E (0.34) KDM4EALDH1A1NPSR1MAPTSMN1; SMN2
SCHEMBL3995952 0.81 KDM4E (0.39) KDM4EALDH1A1NPSR1MAPTSMN1; SMN2
SCHEMBL4117716 0.78 SIGMAR1 (0.33) KDM4EALDH1A1NPSR1MAPTSMN1; SMN2
SCHEMBL8042867 0.77 KDM4E (0.33) KDM4EALDH1A1NPSR1MAPTSMN1; SMN2
SCHEMBL4134627 0.77 MAPT (0.34) KDM4EALDH1A1NPSR1MAPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009071707-A1 NOVEL COMPOUNDS USEFUL FOR THE TREATMENT OF DEGENERATIVE & INFLAMMATORY DISEASES GALAPAGOS NV (BE) 2009-06-11 WO disclosed