SCHEMBL4129431

SCHEMBL4129431

O=C(NCCCOc1cc2cc(S(=O)(=O)NC[PH](=O)O)sc2cc1OCCCC[AsH]C(=O)c1ccc(O)c(O)c1)c1ccc(O)c(O)c1

nearest known ligand 0.37

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
XDH P47989 1/20 0.34
CNR2 P34972 2/20 0.31
SMPD1 P17405 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4155689 0.92 XDH (0.39) XDHCNR2SMPD1
SCHEMBL4565924 0.89 CA2 (0.31)
SCHEMBL3480053 0.81 XDH (0.39) XDHCNR2SMPD1
SCHEMBL3480325 0.81 XDH (0.39) XDHCNR2SMPD1
SCHEMBL3480294 0.78 XDH (0.35) XDHCNR2SMPD1
SCHEMBL4132872 0.75 CNR2 (0.36) XDHCNR2SMPD1
SCHEMBL3480318 0.71 XDH (0.33) XDH
SCHEMBL3480317 0.71 XDH (0.33) XDH
SCHEMBL4138497 0.71 MCL1 (0.36) XDHCNR2SMPD1
SCHEMBL3480605 0.71 TOP1 (0.35) XDHCNR2SMPD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2024376-A1 NOVEL SULFONAMIDOMETHYLPHOSPHONATE INHIBITORS OF BETA-LACTAMASE Merck & Co., Inc. (US) 2009-02-18 EP disclosed
WO-2007139729-A1 NOVEL SULFONAMIDOMETHYLPHOSPHONATE INHIBITORS OF BETA-LACTAMASE MERCK & CO., INC. (US) 2007-12-06 WO disclosed