SCHEMBL4132066

SCHEMBL4132066

Cc1ccc(N=C2NC(=O)C(C(C)c3cccc(C(F)(F)F)c3)S2)cc1

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.45
MAPT P10636 1/20 0.45
HSD11B1 P28845 3/20 0.43
DAO P14920 1/20 0.38
GAA P10253 2/20 0.36
KCNN4 O15554 6/20 0.36
HPGD P15428 1/20 0.35
LMNA P02545 1/20 0.35
NFE2L2 Q16236 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4132065 1.00 TP53 (0.45) TP53MAPTHSD11B1DAOGAA
SCHEMBL4137361 0.89 MAPT (0.44) TP53MAPTHSD11B1DAOGAA
SCHEMBL4132068 0.84 HSD11B1 (0.49) TP53HSD11B1DAOGAAKCNN4
SCHEMBL4130892 0.78 MAPT (0.45) TP53MAPTHSD11B1GAAHPGD
SCHEMBL4130896 0.78 MAPT (0.45) TP53MAPTHSD11B1GAAHPGD
SCHEMBL4136135 0.76 KMT2A (0.57) TP53MAPTGAALMNAALDH1A1
SCHEMBL4136132 0.76 KMT2A (0.57) TP53MAPTGAALMNAALDH1A1
SCHEMBL4137364 0.76 GAA (0.43) TP53MAPTHSD11B1GAALMNA
SCHEMBL4130977 0.74 KMT2A (0.46) TP53MAPTHSD11B1GAALMNA
SCHEMBL4130980 0.74 KMT2A (0.46) TP53MAPTHSD11B1GAALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090156644-A1 Use of thiazole derivatives and analogues in the treatment of cancer BETAGENON AB (SE) 2009-06-18 US disclosed
US-20090136472-A1 Use of thiazole derivatives and analogues in disorders caused by free fatty acids BETAGENON AB (SE) 2009-05-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090156644-A1 Use of thiazole derivatives and analogues in the treatment of cancer TBXA2R, TSHR, FOLR1 TP53 44/4885MAPT 3828/4885HSD11B1 1506/4885
US-20090136472-A1 Use of thiazole derivatives and analogues in disorders caused by free fatty acids FFAR2, FFAR1, FFAR4 TP53 4029/4885MAPT 2648/4885HSD11B1 218/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.