SCHEMBL4132414

SCHEMBL4132414

CC(=O)c1ccc(-c2ccc3c(c2)CCC(N2CCCC2)C3)cc1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.45
FAAH O00519 1/20 0.41
DRD2 P14416 2/20 0.40
DRD3 P35462 2/20 0.40
L3MBTL3 Q96JM7 7/20 0.40
L3MBTL1 Q9Y468 6/20 0.40
MBTD1 Q05BQ5 4/20 0.40
TP53BP1 Q12888 1/20 0.40
L3MBTL4 Q8NA19 1/20 0.40
KDM2B Q8NHM5 2/20 0.39
HTR1D P28221 2/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4128788 0.89 HRH3 (0.49) HRH3FAAHL3MBTL3L3MBTL1
SCHEMBL4136102 0.89 FAAH (0.44) FAAHL3MBTL3L3MBTL1MBTD1TP53BP1
SCHEMBL4132197 0.87 HRH3 (0.53) HRH3FAAHL3MBTL3L3MBTL1
SCHEMBL4143084 0.87 KCNH2 (0.47) HRH3L3MBTL3L3MBTL1KDM2B
SCHEMBL4135538 0.85 L3MBTL3 (0.53) L3MBTL3L3MBTL1MBTD1TP53BP1L3MBTL4
SCHEMBL4135754 0.85 HRH3 (0.42) HRH3FAAHDRD3L3MBTL3KDM2B
SCHEMBL4141827 0.85 HRH3 (0.49) HRH3FAAHKMT2A
SCHEMBL4136657 0.83 HRH3 (0.48) HRH3
SCHEMBL4147479 0.83 FYN (0.44) HRH3FAAHHTR1D
SCHEMBL4144854 0.82 HRH3 (0.52) HRH3MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090163482-A1 TETRALINES ANTAGONISTS OF THE H-3 RECEPTOR MCHARDY STANTON FURST 2009-06-25 US claimed
US-20090163482-A1 TETRALINES ANTAGONISTS OF THE H-3 RECEPTOR MCHARDY STANTON FURST 2009-06-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090163482-A1 TETRALINES ANTAGONISTS OF THE H-3 RECEPTOR HRH3, HRH4, HRH1 HRH3 1/4885FAAH 217/4885DRD2 197/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.