SCHEMBL4134237

SCHEMBL4134237

O=C(O)c1sccc1-c1ccccc1Cl

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RORB Q92753 6/20 0.51
RORC P51449 2/20 0.51
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
BCAT2 O15382 1/20 0.46
PTPRC P08575 2/20 0.46
PTPRG P23470 1/20 0.46
NPSR1 Q6W5P4 2/20 0.44
ALDH1A1 P00352 2/20 0.44
DHODH Q02127 1/20 0.43
KDM4E B2RXH2 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CYP2A6 P11509 1/20 0.41
ALPL P05186 1/20 0.41
GAA P10253 1/20 0.41
PKM P14618 1/20 0.41
MAPK1 P28482 1/20 0.40
MCL1 Q07820 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7472100 0.84 BCAT2 (0.62) RORBRORCKMT2ABCAT2GAA
SCHEMBL953378 0.79 KMT2A (0.52) RORBMEN1KMT2APTPRCPTPRG
SCHEMBL31540411 0.79 BCAT2 (0.46) RORBRORCMEN1KMT2ABCAT2
SCHEMBL31540417 0.79 BCAT2 (0.46) RORBRORCKMT2ABCAT2PTPRC
SCHEMBL16472186 0.79 HPGD (0.51) MEN1KMT2ABCAT2PTPRCNPSR1
SCHEMBL1670982 0.77 BCAT2 (0.72) RORBMEN1KMT2ABCAT2PTPRC
SCHEMBL14397435 0.76 NPSR1 (0.49) RORBRORCBCAT2PTPRCNPSR1
SCHEMBL28910605 0.76 RORC (0.63) RORBRORCMEN1KMT2ABCAT2
Bicarbonate SCHEMBL4865957 0.76 CYP2A6 (0.59) MEN1KMT2APTPRCNPSR1ALDH1A1
Bicarbonate SCHEMBL11009844 0.76 CYP2A6 (0.59) MEN1KMT2APTPRCNPSR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2066675-A1 PROCESS FOR THE PREPARATION OF 4-HYDROXYTHIENO[2,3-B]PYRIDINE-5-CARBONITRILES Wyeth (US) 2009-06-10 EP disclosed
WO-2008039414-A1 PROCESS FOR THE PREPARATION OF 4-HYDROXYTHIENO[2,3-B]PYRIDINE-5-CARBONITRILES WYETH (US) 2008-04-03 WO disclosed