SCHEMBL4143256

SCHEMBL4143256

OCc1ccc(CN2CCOCC2)o1

nearest known ligand 0.61

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.61
CYP2C9 P11712 2/20 0.50
ALOX15 P16050 1/20 0.50
HSD17B10 Q99714 1/20 0.50
HRH3 Q9Y5N1 3/20 0.48
ALDH1A1 P00352 2/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
CXCR4 P61073 1/20 0.44
CYP2A13 Q16696 5/20 0.43
MYC P01106 1/20 0.43
NPSR1 Q6W5P4 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C19 P33261 1/20 0.41
GFER P55789 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11186313 0.88 ALDH1A1 (0.50) HTTALDH1A1MEN1KMT2ANPSR1
SCHEMBL28811140 0.85 KDM4E (0.53) HTTCYP2C9HSD17B10HRH3ALDH1A1
SCHEMBL7329753 0.83 KDM4E (0.55) HTTCYP2C9HSD17B10HRH3ALDH1A1
SCHEMBL4136041 0.81 HTT (0.57) HTTCYP2C9ALOX15HSD17B10HRH3
SCHEMBL13115535 0.81 HTT (0.57) HTTCYP2C9ALOX15HSD17B10HRH3
SCHEMBL11523316 0.80 ALDH1A1 (0.41) HTTALDH1A1MEN1KMT2ANPSR1
SCHEMBL4144775 0.80 ALDH1A1 (0.55) HTTALDH1A1MEN1KMT2ANPSR1
SCHEMBL1472855 0.78 GFER (0.64) HTTCYP2C9ALOX15HSD17B10HRH3
SCHEMBL8263606 0.78 ALDH1A1 (0.63) HTTCYP2C9ALOX15HSD17B10HRH3
SCHEMBL11479737 0.78 HTT (0.57) HTTCYP2C9ALOX15HSD17B10HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019174221-A1 PROCESS FOR PRODUCING AN AMINE IN A SOLVENT SYSTEM CONTAINING WATER RHODIA OPERATIONS (FR) 2019-09-19 WO disclosed
CN-105622554-A Method for preparing 2-hydroxymethyl-5-amine methyl furan compound by fructose DALIAN INST CHEMICAL PHYSICS CAS 2016-06-01 CN disclosed
CN-105503791-A 2-hydroxymethyl-5-aminomethyl-furan compound synthesis method DALIAN INST CHEMICAL PHYSICS CAS 2016-04-20 CN disclosed
US-20090054397-A1 PYRAZOLE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE COMPOUND OHI NORIHITO 2009-02-26 US disclosed
US-20090054397-A1 PYRAZOLE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE COMPOUND OHI NORIHITO 2009-02-26 US disclosed
US-20090054397-A1 PYRAZOLE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE COMPOUND OHI NORIHITO 2009-02-26 US disclosed
US-7429609-B2 Pyrazole compound and medicinal composition containing the same EISAI R & D MANAGEMENT CO., LTD. (JP) 2008-09-30 US disclosed
US-20050261339-A1 Pyrazole compound and medicinal composition containing the same EISAI R&D MANAGEMENT CO., LTD. (JP) 2005-11-24 US disclosed
US-20050208582-A1 Pyrazole compounds and pharmaceutical compositions comprising the compound EISAI R&D MANAGEMENT CO., LTD. (JP) 2005-09-22 US disclosed
CN-1656079-A Pyrazole compounds and pharmaceutical compositions containing the same EISAI CO LTD (JP) 2005-08-17 CN disclosed
EP-1510516-A1 PYRAZOLE COMPOUND AND MEDICINAL COMPOSITION CONTAINING THE SAME Eisai Co., Ltd. (JP) 2005-03-02 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090054397-A1 PYRAZOLE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE COMPOUND CNKSR1, NR3C2, CSNK2B HTT 3425/4885CYP2C9 908/4885ALOX15 3178/4885
US-20050261339-A1 Pyrazole compound and medicinal composition containing the same CNKSR1, NR3C2, CSNK2B HTT 3942/4885CYP2C9 1578/4885ALOX15 3079/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.