SCHEMBL4147293

SCHEMBL4147293

COC(=O)c1cc(C2=C(c3cc(C(F)(F)F)ccc3O)CCC2)cnc1C(F)(F)F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGER1 P34995 3/20 0.42
CYP2C9 P11712 2/20 0.42
CFTR P13569 2/20 0.40
MAPT P10636 1/20 0.39
GAA P10253 1/20 0.37
LMNA P02545 2/20 0.36
PKM P14618 1/20 0.36
TOP2A P11388 1/20 0.36
TLR2 O60603 1/20 0.35
TLR1 Q15399 1/20 0.35
BRAF P15056 1/20 0.33
PDGFRB P09619 1/20 0.33
KDR P35968 1/20 0.33
SLC6A2 P23975 1/20 0.33
MRGPRX4 Q96LA9 1/20 0.33
POLQ O75417 1/20 0.33
POLB P06746 1/20 0.33
TSHR P16473 1/20 0.33
TMPRSS4 Q9NRS4 1/20 0.33
PTGS1 P23219 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4170679 0.90 PTGER1 (0.42) PTGER1CYP2C9CFTRMAPTGAA
SCHEMBL13696751 0.89 PTGER1 (0.43) PTGER1CYP2C9MAPTBRAFMRGPRX4
SCHEMBL4157965 0.89 PTGER1 (0.45) PTGER1CYP2C9MAPTGAALMNA
SCHEMBL4146588 0.79 MAPT (0.41) PTGER1CYP2C9MAPTGAALMNA
SCHEMBL4154455 0.77 CYP2C9 (0.42) PTGER1CYP2C9MAPTGAAMRGPRX4
SCHEMBL4152004 0.75 PTGER1 (0.39) PTGER1CYP2C9CFTRMAPTTOP2A
SCHEMBL13697406 0.74 PTGER1 (0.50) PTGER1CYP2C9MAPTPOLB
SCHEMBL4149095 0.74 PTGER1 (0.54) PTGER1CYP2C9MAPTLMNASLC6A2
SCHEMBL4159517 0.74 PTGER1 (0.64) PTGER1CYP2C9MRGPRX4
SCHEMBL5620094 0.74 CYP2C9 (0.55) PTGER1CYP2C9MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090227591-A1 Cyclopentene compounds GLAXO GROUP LIMITED (GB) 2009-09-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090227591-A1 Cyclopentene compounds C1R, CYP1B1, ADORA2B PTGER1 246/4885CYP2C9 5/4885CFTR 68/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.