SCHEMBL4149031

SCHEMBL4149031

FC(F)(F)c1cccc2[nH]c(-c3cccc4[nH]n[c]c34)nc12

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 4/20 0.49
MGAM O43451 8/20 0.42
GAA P10253 8/20 0.42
SI P14410 8/20 0.42
MGAM2 Q2M2H8 8/20 0.42
PTGES O14684 1/20 0.41
NPY5R Q15761 1/20 0.37
TRPM8 Q7Z2W7 2/20 0.36
CYP2C9 P11712 1/20 0.36
KCNH2 Q12809 1/20 0.36
AXL P30530 1/20 0.35
TRPA1 O75762 2/20 0.34
TRPV1 Q8NER1 1/20 0.34
HDAC3 O15379 1/20 0.34
HDAC7 Q8WUI4 1/20 0.34
HDAC10 Q969S8 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
ATR Q13535 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL558190 0.77 AXL (0.47) PARP1TRPM8AXLTRPA1TRPV1
SCHEMBL1812287 0.75 NPC1 (0.54) GAA
SCHEMBL8818583 0.70 PARP1 (0.63) PARP1MGAMGAASIMGAM2
SCHEMBL505343 0.70 DHODH (0.57) PARP1MGAMGAASIMGAM2
SCHEMBL183317 0.69 METAP2 (0.48) NPY5R
SCHEMBL12934190 0.68 PARP1 (0.50) PARP1GAAPTGESNPY5RAXL
SCHEMBL31027935 0.68 HDAC6 (0.58) PARP1MGAMGAASIMGAM2
SCHEMBL22452437 0.68 HDAC6 (0.58) PARP1MGAMGAASIMGAM2
SCHEMBL124272 0.68 CBFB (0.68)
SCHEMBL1889612 0.67 PARP1 (0.80) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8080573-B2 Heterocycle substituted amide and sulfur amide derivatives as histone deacetylase (hdac) inhibitors ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2011-12-20 US disclosed
US-20090156619-A1 Heterocycle Substituted Amide and Sulfur Amide Derivatives as Histone Deacetylase (HDAC) Inhibitors MSD ITALIA S.R.L. (IT) 2009-06-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090156619-A1 Heterocycle Substituted Amide and Sulfur Amide Derivatives as Histone Deacetylase (HDAC) Inhibitors HDAC1, HDAC6, HDAC11 PARP1 959/4885MGAM 4236/4885GAA 705/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.