SCHEMBL4149979

SCHEMBL4149979

O=C(Nc1ccc(NC(=O)c2ccnc3[nH]c(-c4ccccc4)nc23)cc1)c1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRMT5 O14744 1/20 0.57
MMP2 P08253 5/20 0.55
MMP9 P14780 5/20 0.55
MMP8 P22894 5/20 0.55
MMP13 P45452 5/20 0.55
HPSE Q9Y251 1/20 0.50
NR2E3 Q9Y5X4 1/20 0.50
PTPN1 P18031 3/20 0.48
AURKA O14965 1/20 0.47
MAPK13 O15264 1/20 0.47
CHEK2 O96017 1/20 0.47
NTRK1 P04629 1/20 0.47
RET P07949 1/20 0.47
HCK P08631 1/20 0.47
FGFR1 P11362 1/20 0.47
FLT4 P35916 1/20 0.47
LIMK1 P53667 1/20 0.47
SIK1 P57059 1/20 0.47
TNK2 Q07912 1/20 0.47
AURKB Q96GD4 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4152155 0.93 GSK3B (0.48) PRMT5MMP2MMP9MMP8MMP13
SCHEMBL4161603 0.89 PRMT5 (0.48) PRMT5MMP2MMP9MMP8MMP13
SCHEMBL13778063 0.88 GSK3B (0.55) PRMT5MMP2MMP9MMP8MMP13
SCHEMBL4152144 0.85 GSK3B (0.60) PRMT5MMP2MMP9MMP8MMP13
SCHEMBL4152662 0.83 RAB9A (0.54) POLBJAK2
SCHEMBL4145718 0.81 DHODH (0.57)
SCHEMBL4153576 0.79 DHODH (0.43) PRMT5MMP2MMP9MMP8MMP13
SCHEMBL4144903 0.79 RAD52 (0.46) PRMT5MMP2MMP9MMP8MMP13
SCHEMBL17224889 0.78 DHODH (0.62)
SCHEMBL4157245 0.78 MMP2 (0.52) PRMT5MMP2MMP9MMP8MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090170847-A1 Imidazopyridine Derivatives Inhibiting Protein Kinase Activity, Method for the Preparation Thereof and Pharmaceutical Composition Containing Same YUYU PHARMA, INC. (KR) 2009-07-02 US claimed
EP-1984370-A1 IMIDAZOPYRIDINE DERIVATIVES INHIBITING PROTEIN KINASE ACTIVITY, METHOD FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITION CONTAINING SAME Crystalgenomics, Inc. (KR) 2008-10-29 EP claimed
WO-2007083978-A1 IMIDAZOPYRIDINE DERIVATIVES INHIBITING PROTEIN KINASE ACTIVITY, METHOD FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITION CONTAINING SAME CRYSTALGENOMICS, INC. (KR) 2007-07-26 WO claimed
US-20090170847-A1 Imidazopyridine Derivatives Inhibiting Protein Kinase Activity, Method for the Preparation Thereof and Pharmaceutical Composition Containing Same YUYU PHARMA, INC. (KR) 2009-07-02 US disclosed
US-20090170847-A1 Imidazopyridine Derivatives Inhibiting Protein Kinase Activity, Method for the Preparation Thereof and Pharmaceutical Composition Containing Same YUYU PHARMA, INC. (KR) 2009-07-02 US disclosed
US-20090170847-A1 Imidazopyridine Derivatives Inhibiting Protein Kinase Activity, Method for the Preparation Thereof and Pharmaceutical Composition Containing Same YUYU PHARMA, INC. (KR) 2009-07-02 US disclosed
WO-2007083978-A1 IMIDAZOPYRIDINE DERIVATIVES INHIBITING PROTEIN KINASE ACTIVITY, METHOD FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITION CONTAINING SAME CRYSTALGENOMICS, INC. (KR) 2007-07-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090170847-A1 Imidazopyridine Derivatives Inhibiting Protein Kinase Activity, Method for the Preparation Thereof and Pharmaceutical Composition Containing Same GSK3B, GSK3A, MAP3K3 PRMT5 882/4885MMP2 1673/4885MMP9 1404/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.