SCHEMBL4150276

SCHEMBL4150276

Nc1cc(-c2ccsc2)nc2ccccc12

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.68
NCF1 P14598 1/20 0.47
TACR3 P29371 1/20 0.46
PDGFRB P09619 1/20 0.45
PDGFRA P16234 1/20 0.45
CYP2E1 P05181 1/20 0.43
CYP2A6 P11509 1/20 0.43
CYP2B6 P20813 1/20 0.43
NPC1 O15118 1/20 0.42
TOP1 P11387 2/20 0.42
CHRNA7 P36544 1/20 0.41
HTR3A P46098 1/20 0.41
KCNH2 Q12809 1/20 0.41
BACE1 P56817 1/20 0.41
NQO2 P16083 1/20 0.41
ADORA2A P29274 2/20 0.40
ADORA1 P30542 2/20 0.40
GBA1 P04062 1/20 0.40
ATR Q13535 1/20 0.40
LMNA P02545 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2873300 0.81 ACHE (1.00) ACHENCF1KCNH2NQO2ADORA2A
SCHEMBL10608842 0.81 TACR3 (0.49) ACHETACR3PDGFRBPDGFRACYP2E1
SCHEMBL6534319 0.81 TACR3 (0.46) ACHETACR3PDGFRBPDGFRACYP2E1
SCHEMBL24505991 0.79 ACHE (0.80) ACHENCF1NPC1ADORA2AADORA1
SCHEMBL28516025 0.78 ACHE (0.93) ACHENCF1ADORA2AADORA1LMNA
SCHEMBL13957916 0.78 KDM4E (0.70) TACR3NPC1LMNASMN1; SMN2KDM4E
Oxalic Acid SCHEMBL1062152 0.74 ACHE (0.83) ACHENCF1TACR3KCNH2ADORA2A
SCHEMBL15919363 0.74 ACHE (0.77) ACHENCF1LMNASMN1; SMN2KDM4E
SCHEMBL4143397 0.74 ACHE (0.77) ACHENCF1NPC1ADORA2AADORA1
SCHEMBL4155489 0.74 ACHE (0.72) ACHENCF1NPC1ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090069338-A1 Method for predicting skin sensitizing activity of compounds DICKSON JR JOHN K 2009-03-12 US disclosed
US-7452887-B2 Quinoline- and isoquinoline-based compounds exhibiting ATP-utilizing enzyme inhibitory activity, and compositions, and uses thereof AMPHORA DISCOVERY CORPORATION (US) 2008-11-18 US disclosed
US-20060009460-A1 Quinoline- and isoquinoline-based compounds exhibiting ATP-utilizing enzyme inhibitory activity, and compositions, and uses thereof AGRIUS GROUP, LLC. 2006-01-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090069338-A1 Method for predicting skin sensitizing activity of compounds ATP5ME, ABCG2, ATP5MG ACHE 31/4885NCF1 672/4885TACR3 2500/4885
US-20060009460-A1 Quinoline- and isoquinoline-based compounds exhibiting ATP-utilizing enzyme inhibitory activity, and compositions, and uses thereof ATP5ME, ATP5MG, ATP5MK ACHE 12/4885NCF1 2180/4885TACR3 2602/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.