SCHEMBL4151724

SCHEMBL4151724

N[C@@H](CCCSCC(=O)C(F)(F)F)C(=O)NCc1cnc2ccccc2c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 2/20 0.41
TPH1 P17752 1/20 0.40
CES1 P23141 1/20 0.39
ATG4B Q9Y4P1 1/20 0.38
GLS O94925 1/20 0.38
NLN Q9BYT8 1/20 0.38
HDAC1 Q13547 2/20 0.37
HDAC2 Q92769 2/20 0.37
CYP1A2 P05177 1/20 0.37
MMP1 P03956 1/20 0.36
FCER2 P06734 1/20 0.36
MMP3 P08254 1/20 0.36
MMP9 P14780 1/20 0.36
OPRK1 P41145 2/20 0.35
HDAC3 O15379 1/20 0.35
HDAC4 P56524 1/20 0.35
HDAC7 Q8WUI4 1/20 0.35
HDAC10 Q969S8 1/20 0.35
HDAC11 Q96DB2 1/20 0.35
HDAC8 Q9BY41 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4151722 0.83 SIRT2 (0.41) MCHR1TPH1CES1ATG4BGLS
Trifluoroacetic Acid SCHEMBL4156590 0.81 SIRT2 (0.41) MCHR1TPH1CES1GLSHDAC1
Trifluoroacetic Acid SCHEMBL4163740 0.79 MCHR1 (0.41) MCHR1CES1ATG4BHDAC1HDAC2
Trifluoroacetic Acid SCHEMBL4166172 0.78 SIRT2 (0.41) MCHR1TPH1CES1GLSHDAC1
Trifluoroacetic Acid SCHEMBL4166154 0.77 SIRT2 (0.38) MCHR1TPH1CES1HDAC1HDAC2
Trifluoroacetic Acid SCHEMBL4162610 0.77 HDAC1 (0.34) MCHR1TPH1CES1HDAC1HDAC2
Trifluoroacetic Acid SCHEMBL4165163 0.75 SIRT2 (0.38) MCHR1TPH1CES1GLSHDAC1
SCHEMBL4156445 0.75 CES1 (0.59) CES1HDAC1HDAC2HDAC3HDAC4
Trifluoroacetic Acid SCHEMBL4151859 0.75 MCHR1 (0.42) MCHR1GLSHDAC1CYP1A2
Trifluoroacetic Acid SCHEMBL4162623 0.75 SIRT2 (0.38) MCHR1TPH1CES1GLSHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090054448-A1 Amino Acid Derivatives as Histone Deacetylase (HDAC) Inhibitors JONES PHILIP 2009-02-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090054448-A1 Amino Acid Derivatives as Histone Deacetylase (HDAC) Inhibitors HDAC5, HDAC1, HDAC11 MCHR1 3532/4885TPH1 101/4885CES1 1925/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.