SCHEMBL4152232

SCHEMBL4152232

O=C(O)C1(c2ccccc2)CCC2(CC1)OCCO2.O=C=NC1(c2ccccc2)CCC2(CC1)OCCO2

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C1 Q04828 1/20 0.45
KMT2A Q03164 3/20 0.36
TET3 O43151 1/20 0.36
FBXL19 Q6PCT2 1/20 0.36
CXXC5 Q7LFL8 1/20 0.36
TET1 Q8NFU7 1/20 0.36
KDM2B Q8NHM5 1/20 0.36
CXXC4 Q9H2H0 1/20 0.36
KDM2A Q9Y2K7 1/20 0.36
ALDH1A1 P00352 4/20 0.36
ALOX15 P16050 1/20 0.35
HSD11B1 P28845 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.34
MEN1 O00255 1/20 0.34
NPC1 O15118 1/20 0.34
MAPK1 P28482 1/20 0.34
CASP1 P29466 1/20 0.34
RAB9A P51151 1/20 0.34
CASP7 P55210 1/20 0.34
HSD17B10 Q99714 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL736092 0.89 POLB (0.39) KMT2AALDH1A1SMN1; SMN2MEN1NPC1
SCHEMBL735386 0.85 AKR1C1 (0.61) AKR1C1KMT2ATET3FBXL19CXXC5
SCHEMBL4152236 0.81 ALDH1A1 (0.34) KMT2AALDH1A1SMN1; SMN2MEN1NPC1
SCHEMBL3134616 0.77 MEN1 (0.38) AKR1C1KMT2AMEN1HDAC4
SCHEMBL23248029 0.73 ALDH1A1 (0.39) KMT2AALDH1A1ALOX15SMN1; SMN2MEN1
SCHEMBL3219496 0.72 APP (0.50) AKR1C1KMT2AHSD11B1NPC1RAB9A
SCHEMBL31016196 0.72 AKR1C1 (0.83) AKR1C1KMT2ATET3FBXL19CXXC5
SCHEMBL6391 0.72 AKR1C1 (0.83) AKR1C1KMT2ATET3FBXL19CXXC5
SCHEMBL1313846 0.70 AKR1C1 (0.42) AKR1C1HDAC4
SCHEMBL4322724 0.70 AKR1C1 (0.38) AKR1C1KMT2AHSD11B1MEN1HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2044016-A2 4-HETEROARYL-SUBSTITUTED 1-AMINOCYCLOHEXANE-1-AND CYCLOHEXENE-1-DERIVATIVES HAVING EFFECTS ON THE OPIOD RECEPTOR SYSTEM Grünenthal GmbH (DE) 2009-04-08 EP disclosed
WO-2008009415-A2 4-HETEROARYL-SUBSTITUTED 1-AMINOCYCLOHEXANE-1- AND CYCLOHEXENE-1-DERIVATIVES HAVING EFFECTS ON THE OPIOD RECEPTOR SYSTEM Grünenthal GmbH (DE) 2008-01-24 WO disclosed