Suxamethonium

Suxamethonium

SCHEMBL41537

C[N+](C)(C)CCOC(=O)CCC(=O)OCC[N+](C)(C)C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

CHRNA1CHRNB1CHRNDCHRNECHRNG

The experimentally established mechanism targets of Suxamethonium. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 1/20 1.00
ADRA1A P35348 1/20 1.00
MAPT P10636 1/20 0.95
BLM P54132 1/20 0.95
CYP2C19 P33261 2/20 0.67
CHRM1 P11229 8/20 0.65
CHRM3 P20309 8/20 0.65
CHRM2 P08172 7/20 0.65
CHRM4 P08173 7/20 0.65
CHRM5 P08912 6/20 0.65
CHRNB2 P17787 4/20 0.65
CHRNA4 P43681 4/20 0.65
CHRNA7 P36544 3/20 0.65
HTR1A P08908 2/20 0.65
SMN1; SMN2 Q16637 2/20 0.65
PGR P06401 1/20 0.65
TBXA2R P21731 1/20 0.65
CHRNB4 P30926 1/20 0.65
CHRNA3 P32297 1/20 0.65
CHRNA10 Q9GZZ6 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Suxamethonium SCHEMBL41536 0.97 MAPT (1.00) ADRA2AADRA1AMAPTBLMCYP2C19
Suxamethonium SCHEMBL2690356 0.97 ADRA2A (0.95) ADRA2AADRA1AMAPTBLMCYP2C19
Suxamethonium SCHEMBL21356923 0.97 ADRA2A (0.95) ADRA2AADRA1AMAPTBLMCYP2C19
Suxamethonium SCHEMBL16320883 0.97 ADRA2A (0.95) ADRA2AADRA1AMAPTBLMCYP2C19
Suxamethonium SCHEMBL1643328 0.97 ADRA2A (0.95) ADRA2AADRA1AMAPTBLMCYP2C19
Suxamethonium SCHEMBL2821312 0.97 ADRA2A (0.95) ADRA2AADRA1AMAPTBLMCYP2C19
Suxamethonium SCHEMBL20815392 0.95 MAPT (0.95) ADRA2AADRA1AMAPTBLMCYP2C19
Suxamethonium SCHEMBL1983256 0.95 MAPT (0.95) ADRA2AADRA1AMAPTBLMCYP2C19
SCHEMBL12560604 0.91 ADRA2A (0.83) ADRA2AADRA1AMAPTBLMCYP2C19
SCHEMBL357905 0.91 ADRA2A (0.83) ADRA2AADRA1AMAPTBLMCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 9705 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4719552-A1 INDUCTION OF GENERAL ANESTHESIA IN ADULTS UNDERGOING ELECTIVE SURGERY Xizang Haisco Pharmaceutical Co., Ltd. (CN) 2026-04-08 EP claimed
EP-4076560-B1 SURFACE MODIFYING COATING FOR MEDICAL DEVICES HOSPIRA INC (US) 2026-04-01 EP claimed
EP-4221200-B1 DEVICE AND METHOD FOR CODING VIDEO DATA BASED ON ONE OR MORE REFERENCE LINES SHARP KK (JP) 2026-03-04 EP claimed
US-20260000678-A1 PHARMACEUTICAL COMPOSITION FOR PREVENTING, SUPPRESSING, OR TREATING SYMPTOM ASSOCIATED WITH PSEUDO-ALLERGIC REACTION TAKASAKI UNIV OF HEALTH AND WELFARE (JP) 2026-01-01 US claimed
EP-4655448-A1 OBJECT, METHOD FOR FUNCTIONALIZING AN OBJECT AND OBJECT WHICH CAN BE OBTAINED THEREFROM, AND METHOD FOR BINDING A PEPTIDE, AND USE OF AN OBJECT FOR BINDING A PEPTIDE Wenatex Forschung - Entwicklung - Produktion GmbH (AT) 2025-12-03 EP claimed
US-12403262-B2 Tamper evident assembly with RFID for syringes FRESENIUS KABI USA, LLC (US) 2025-09-02 US claimed
US-20250249185-A1 TAMPER EVIDENT CAP WITH RFID FOR SYRINGES FRESENIUS KABI USA, LLC 2025-08-07 US claimed
US-20250243208-A1 BICYCLIC HETEROCYCLES AS MRGPRX2 ANTAGONISTS INCYTE CORPORATION 2025-07-31 US claimed
EP-4249494-B1 A DRUG COMPRISING A RADICAL GENERATING CATALYST ACENET INC (JP) 2025-07-16 EP claimed
US-20250206734-A1 BICYCLIC HETEROCYCLES AS MRGPRX2 ANTAGONISTS INCYTE CORPORATION 2025-06-26 US claimed
EP-0575479-A1 PRODUCTION AND USE OF BUTYRYLCHOLINESTERASE PHARMAVENE, INC. (US) 1993-12-29 EP claimed
WO-1993001830-A1 EXPRESSION OF ENZYMATICALLY ACTIVE RECOMBINANT HUMAN ACETYLCHOLINESTERASE AND USES THEREOF BIO-TECHNOLOGY GENERAL CORP. (US) 1993-02-04 WO claimed
WO-1992014483-A1 PRODUCTION AND USE OF BUTYRYLCHOLINESTERASE PHARMAVENE, INC. (US) 1992-09-03 WO claimed
EP-0126684-B1 DRUG DELIVERY SYSTEM UTILIZING THERMOSETTING GELS MERCK & CO. INC. (US) 1991-08-28 EP claimed
EP-0388906-A2 Genetically engineered human cholinesterases YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM (IL) 1990-09-26 EP claimed
US-4726594-A Drug injection system for use with an arrow BENKE GUS A (US) 1988-02-23 US claimed
EP-0206200-A2 Human cholinesterase-type proteins and their production YEDA RESEARCH AND DEVELOPMENT COMPANY LIMITED (IL) 1986-12-30 EP claimed
EP-0147780-A2 Drug delivery device MERCK & CO. INC. (US) 1985-07-10 EP claimed
EP-0126684-A2 Drug delivery system utilizing thermosetting gels MERCK & CO. INC. (US) 1984-11-28 EP claimed
US-4474752-A DIAMINE MODIFIED POLYOXYETHYLENE-POLYOXYPROPYLENE COPOLYMER MERCK & CO., INC. (US) 1984-10-02 US claimed