SCHEMBL4155171

SCHEMBL4155171

NN(c1ccccc1)c1ncccn1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.39
NOS1 P29475 1/20 0.39
NOS2 P35228 1/20 0.39
PI4KA P42356 1/20 0.39
PI4K2B Q8TCG2 1/20 0.39
PI4K2A Q9BTU6 1/20 0.39
PI4KB Q9UBF8 1/20 0.39
USP2 O75604 1/20 0.38
KDM4E B2RXH2 5/20 0.37
GAA P10253 1/20 0.37
CYP1A2 P05177 2/20 0.36
LMNA P02545 2/20 0.36
P4HTM Q9NXG6 2/20 0.36
POLB P06746 1/20 0.36
CCR1 P32246 1/20 0.36
CCR5 P51681 1/20 0.36
CCR8 P51685 1/20 0.36
METAP1 P53582 1/20 0.36
BLM P54132 1/20 0.36
HIF1A Q16665 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3394969 0.84 HSP90AA1 (0.33) KDM4EGAACYP1A2ALDH1A1TDP1
SCHEMBL7511419 0.82 ALDH1A1 (0.41) KDM4ECYP1A2LMNAALDH1A1TDP1
SCHEMBL3361750 0.79 ALDH1A1 (0.42) NOS3NOS1NOS2PI4KAPI4K2B
Hydrochloric Acid SCHEMBL1718427 0.78 ALDH1A1 (0.42) KDM4EGAACYP1A2ALDH1A1TDP1
SCHEMBL193916 0.78 ALDH1A1 (0.46) KDM4EGAACYP1A2ALDH1A1TDP1
SCHEMBL1792016 0.78 ALDH1A1 (0.46) KDM4EGAACYP1A2ALDH1A1TDP1
Hydrochloric Acid SCHEMBL250009 0.75 ALDH1A1 (0.43) KDM4EGAACYP1A2BLMALDH1A1
Ammonia Solution, Strong SCHEMBL28763213 0.75 ALDH1A1 (0.43) KDM4EGAACYP1A2ALDH1A1TDP1
Ammonia Solution, Strong SCHEMBL28873134 0.75 ALDH1A1 (0.43) KDM4EGAACYP1A2ALDH1A1TDP1
Water SCHEMBL8817645 0.75 ALDH1A1 (0.43) KDM4EGAACYP1A2ALDH1A1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104109127-B Kinase inhibitor and the method for treating related disease 北京大学深圳研究生院 2019-11-05 CN disclosed
CN-104109127-B Kinase inhibitor and the method for treating related disease 北京大学深圳研究生院 2019-11-05 CN disclosed
CN-109305944-A The inhibitor of bruton's tyrosine kinase 深圳睿熙生物科技有限公司 2019-02-05 CN disclosed
CN-103073508-B The method of inhibitors of kinases and treatment relevant disease PEKING UNIVERSITY SHENZHEN GRADUATE SCHOOL (CN) 2016-06-01 CN disclosed
CN-103073508-B The method of inhibitors of kinases and treatment relevant disease PEKING UNIVERSITY SHENZHEN GRADUATE SCHOOL (CN) 2016-06-01 CN disclosed
CN-102066339-A 2, 6-diamino-pyrimidin-5-yl-carboxamides as SYK or JAK protein kinase inhibitors PORTOLA PHARM INC 2011-05-18 CN disclosed
US-20090240035-A1 DNA REPLICATION PROTEINS OF GRAM POSITIVE BACTERIA AND THEIR USE TO SCREEN FOR CHEMICAL INHIBITORS O'DONNELL MICHAEL E 2009-09-24 US disclosed
US-7557184-B2 Isolated staphylococcus DNAX subunit and use thereof THE ROCKEFELLER UNIVERSITY (US) 2009-07-07 US disclosed
US-20090123911-A9 ISOLATED STAPHYLOCOCCUS DNAX SUBUNIT AND USE THEREOF O'DONNELL MICHAEL E 2009-05-14 US disclosed
US-20090004675-A1 Method of Identifying Compounds for Bacterial Growth Modulation THE ROCKEFELLER UNIVERSITY (US) 2009-01-01 US disclosed
US-7432365-B1 DNA molecules encoding beta clamp proteins of gram positive bacteria THE ROCKEFELLER UNIVERSITY 2008-10-07 US disclosed
WO-2006052746-A2 METHOD OF IDENTIFYING COMPOUNDS FOR BACTERIAL GROWTH MODULATION THE ROCKEFELLER UNIVERSITY (US) 2006-05-18 WO disclosed
US-20030129633-A1 DNA replication proteins of Gram positive bacteria and their use to screen for chemical inhibitors O'DONNELL MICHAEL E (US) 2003-07-10 US disclosed
EP-1056763-A4 DNA REPLICATION PROTEINS OF GRAM POSITIVE BACTERIA AND THEIR USE TO SCREEN FOR CHEMICAL INHIBITORS UNIV ROCKEFELLER (US) 2003-03-26 EP disclosed
WO-2001009164-A2 DNA REPLICATION PROTEINS OF GRAM POSITIVE BACTERIA AND THEIR USE TO SCREEN FOR CHEMICAL INHIBITORS THE ROCKEFELLER UNIVERSITY (US) 2001-02-08 WO disclosed
EP-1056763-A1 DNA REPLICATION PROTEINS OF GRAM POSITIVE BACTERIA AND THEIR USE TO SCREEN FOR CHEMICAL INHIBITORS THE ROCKEFELLER UNIVERSITY (US) 2000-12-06 EP disclosed
WO-1999037661-A9 DNA REPLICATION PROTEINS OF GRAM POSITIVE BACTERIA AND THEIR USE TO SCREEN FOR CHEMICAL INHIBITORS UNIV ROCKEFELLER (US) 1999-12-02 WO disclosed
WO-1999037661-A1 DNA REPLICATION PROTEINS OF GRAM POSITIVE BACTERIA AND THEIR USE TO SCREEN FOR CHEMICAL INHIBITORS THE ROCKEFELLER UNIVERSITY (US) 1999-07-29 WO disclosed