SCHEMBL4159624

SCHEMBL4159624

N[C@@H](CCCSCC(=O)C(F)(F)F)C(=O)N(CCc1ccccc1)C(=O)Cc1ccsc1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CES1 P23141 6/20 0.47
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
OPRM1 P35372 2/20 0.35
OPRD1 P41143 2/20 0.35
OPRK1 P41145 2/20 0.35
FAAH O00519 3/20 0.33
RAB9A P51151 1/20 0.32
GRIK1 P39086 1/20 0.31
SLC1A3 P43003 2/20 0.31
SLC1A2 P43004 2/20 0.31
SLC1A1 P43005 2/20 0.31
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4159627 0.84 CES1 (0.47) CES1HDAC1HDAC2OPRM1OPRD1
Trifluoroacetic Acid SCHEMBL4169493 0.78 CES1 (0.34) CES1HDAC1HDAC2
SCHEMBL4173031 0.78 POLB (0.32) CES1POLB
Trifluoroacetic Acid SCHEMBL4160625 0.75 CES1 (0.38) CES1HDAC1HDAC2FAAHRAB9A
SCHEMBL4162818 0.75 CES1 (0.43) CES1HDAC1HDAC2POLB
SCHEMBL4605724 0.73 CES1 (0.46) CES1HDAC1HDAC2OPRM1OPRD1
SCHEMBL4171426 0.72 CES1 (0.44) CES1HDAC1HDAC2FAAH
SCHEMBL4606140 0.72 CES1 (0.35) CES1HDAC1HDAC2OPRM1
SCHEMBL4156445 0.71 CES1 (0.59) CES1HDAC1HDAC2FAAHPOLB
SCHEMBL4174427 0.71 SIGMAR1 (0.36) CES1HDAC1HDAC2OPRM1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090054448-A1 Amino Acid Derivatives as Histone Deacetylase (HDAC) Inhibitors JONES PHILIP 2009-02-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090054448-A1 Amino Acid Derivatives as Histone Deacetylase (HDAC) Inhibitors HDAC5, HDAC1, HDAC11 CES1 1925/4885HDAC1 2/4885HDAC2 7/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.