SCHEMBL4162402

SCHEMBL4162402

CCC(Br)(C(N)=O)c1ccccn1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BLM P54132 2/20 0.45
SLC22A2 O15244 1/20 0.45
SLC22A1 O15245 1/20 0.45
PGR P06401 1/20 0.45
THRB P10828 1/20 0.45
ADRB3 P13945 1/20 0.45
OPRK1 P41145 1/20 0.45
PMP22 Q01453 1/20 0.45
KCNH2 Q12809 1/20 0.45
PDE3A Q14432 1/20 0.45
SLC47A1 Q96FL8 1/20 0.45
CYP3A4 P08684 1/20 0.45
ALOX15 P16050 1/20 0.45
TSHR P16473 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
SMN1; SMN2 Q16637 2/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
NOS3 P29474 2/20 0.43
NOS1 P29475 2/20 0.43
NOS2 P35228 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3743980 0.85 L3MBTL1 (0.46) BLMSLC22A2SLC22A1PGRTHRB
SCHEMBL666125 0.80 BLM (0.45) BLMSLC22A2SLC22A1PGRTHRB
SCHEMBL3954412 0.79 BLM (0.44) BLMSLC22A2SLC22A1PGRTHRB
SCHEMBL4036415 0.76 BLM (0.42) BLMSLC22A2SLC22A1PGRTHRB
SCHEMBL4030399 0.76 BLM (0.42) BLMSLC22A2SLC22A1PGRTHRB
SCHEMBL2700564 0.76 TDP1 (0.42) BLMSLC22A2SLC22A1PGRTHRB
SCHEMBL2465434 0.75 SMN1; SMN2 (0.50) BLMSLC22A2SLC22A1PGRTHRB
SCHEMBL8283520 0.75 MAPT (0.52) BLMSLC22A2SLC22A1PGRTHRB
SCHEMBL18766023 0.75 BLM (0.44) BLMSLC22A2SLC22A1PGRTHRB
SCHEMBL3138017 0.74 MAPT (0.55) KCNH2LMNACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010493-A2 PYRIDYL AMIDE T-TYPE CALCIUM CHANNEL ANTAGONISTS Merck & Co., Inc. (US) 2009-01-07 EP disclosed
WO-2007120729-A2 PYRIDYL AMIDE T-TYPE CALCIUM CHANNEL ANTAGONISTS MERCK & CO., INC. (US) 2007-10-25 WO disclosed