SCHEMBL4162702

SCHEMBL4162702

CC(OCC1(Cc2ccc(F)cc2)CCNCC1)c1cc(Cl)cc2cn(CC3CC3)nc12

nearest known ligand 0.33

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 1/20 0.33
TACR1 P25103 1/20 0.31
SLC6A4 P31645 1/20 0.31
KCNH2 Q12809 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4162696 1.00 TGFBR1 (0.33) TGFBR1TACR1SLC6A4KCNH2
SCHEMBL12289964 0.87 TACR1 (0.42) TGFBR1TACR1SLC6A4KCNH2
SCHEMBL4442401 0.82 TGFBR1 (0.31) TGFBR1SLC6A4
SCHEMBL4442397 0.82 TGFBR1 (0.31) TGFBR1SLC6A4
SCHEMBL2426694 0.79 TACR1 (0.43) TACR1SLC6A4KCNH2
SCHEMBL2426692 0.79 TACR1 (0.43) TACR1SLC6A4KCNH2
SCHEMBL3932352 0.77 TACR1 (0.36) TACR1SLC6A4KCNH2
SCHEMBL13961177 0.76 TACR1 (0.43) TACR1SLC6A4KCNH2
SCHEMBL2428697 0.75 TACR1 (0.31) TACR1SLC6A4KCNH2
SCHEMBL3935770 0.75

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009009411-A1 SUBSTITUTED HETEROCYCLIC ETHERS AND THEIR USE IN CNS DISORDERS BRISTOL-MYERS SQUIBB COMPANY (US) 2009-01-15 WO claimed
WO-2009009411-A1 SUBSTITUTED HETEROCYCLIC ETHERS AND THEIR USE IN CNS DISORDERS BRISTOL-MYERS SQUIBB COMPANY (US) 2009-01-15 WO disclosed