SCHEMBL4442397

SCHEMBL4442397

C[C@@H](OCC1(Cc2ccc(F)cc2)CCNCC1)c1cc(Cl)cc2cnn(CC3CC3)c12

nearest known ligand 0.32

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 1/20 0.31
HTR2A P28223 1/20 0.30
HTR2C P28335 1/20 0.30
SLC6A4 P31645 1/20 0.30
ALK Q9UM73 1/20 0.30
JAK2 O60674 1/20 0.30
JAK1 P23458 1/20 0.30
TYK2 P29597 1/20 0.30
JAK3 P52333 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4442401 1.00 TGFBR1 (0.31) TGFBR1HTR2AHTR2CSLC6A4ALK
SCHEMBL4162696 0.82 TGFBR1 (0.33) TGFBR1SLC6A4
SCHEMBL4162702 0.82 TGFBR1 (0.33) TGFBR1SLC6A4
SCHEMBL2429710 0.79 TACR1 (0.41) SLC6A4
SCHEMBL2429709 0.79 TACR1 (0.41) SLC6A4
SCHEMBL12290816 0.74 TACR1 (0.40) SLC6A4
SCHEMBL2425778 0.74 TP53 (0.38)
SCHEMBL2425779 0.74 TP53 (0.38)
SCHEMBL2428697 0.72 TACR1 (0.31) SLC6A4
SCHEMBL2429202 0.70 TACR1 (0.42) SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009009411-A1 SUBSTITUTED HETEROCYCLIC ETHERS AND THEIR USE IN CNS DISORDERS BRISTOL-MYERS SQUIBB COMPANY (US) 2009-01-15 WO disclosed