SCHEMBL4164895

SCHEMBL4164895

Brc1cnc2[nH]ncc2c1N1CCNCC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.54
CHEK2 O96017 1/20 0.54
AURKA O14965 2/20 0.41
CHRNB2 P17787 4/20 0.40
CHRNA4 P43681 4/20 0.40
PLK4 O00444 1/20 0.40
PAK4 O96013 1/20 0.40
HSP90AA1 P07900 1/20 0.39
HSP90AB1 P08238 1/20 0.39
ADRB2 P07550 1/20 0.39
AKT2 P31751 2/20 0.38
PIK3CD O00329 1/20 0.38
PIK3CA P42336 1/20 0.38
PIK3CB P42338 1/20 0.38
HTR2B P41595 2/20 0.36
HTR6 P50406 2/20 0.36
HTR1A P08908 1/20 0.36
HTR7 P34969 1/20 0.36
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3718343 0.98 CHEK1 (0.53) CHEK1CHEK2AURKACHRNB2CHRNA4
Hydrochloric Acid SCHEMBL3720255 0.81 PLK4 (0.44) CHEK1CHEK2PLK4PAK4ADRB2
Hydrochloric Acid SCHEMBL3723324 0.81 ADRB2 (0.53) CHEK1CHEK2CHRNB2CHRNA4PLK4
SCHEMBL3718717 0.78 EPHX2 (0.43) CHEK1CHEK2PLK4PAK4ADRB2
SCHEMBL3736680 0.78 AKT2 (0.41) CHEK1CHEK2PLK4PAK4ADRB2
SCHEMBL3721308 0.78 HTR2C (0.55) AURKACHRNB2CHRNA4HTR6HTR2C
Hydrochloric Acid SCHEMBL3716007 0.77 ROCK2 (0.42) CHEK1CHEK2PLK4PAK4ADRB2
Hydrochloric Acid SCHEMBL3713877 0.77 ADRB2 (0.43) CHEK1CHEK2PLK4PAK4ADRB2
Hydrochloric Acid SCHEMBL3721311 0.77 AKT2 (0.40) CHEK1CHEK2PLK4PAK4ADRB2
Hydrochloric Acid SCHEMBL3721934 0.77 AKT2 (0.40) CHEK1CHEK2PLK4PAK4ADRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009089359-A1 PYRAZOLOPYRIDINES AS KINASE INHIBITORS ARRAY BIOPHARMA INC. (US) 2009-07-16 WO disclosed