Enilconazole

Enilconazole

SCHEMBL41653

C=CCOC(Cn1ccnc1)c1ccc(Cl)cc1Cl.O=S(=O)(O)O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

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

The experimentally established mechanism targets of Enilconazole. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB1 known ✓ P08588 3/20 0.64
SLC6A2 known ✓ P23975 3/20 0.64
OPRK1 known ✓ P41145 3/20 0.64
SLC6A3 known ✓ Q01959 3/20 0.64
CHRM2 known ✓ P08172 2/20 0.64
ADRA2A known ✓ P08913 2/20 0.64
CHRM1 known ✓ P11229 2/20 0.64
ADRB3 known ✓ P13945 2/20 0.64
ADRA2B known ✓ P18089 2/20 0.64
CHRM3 known ✓ P20309 2/20 0.64
ADRA1D known ✓ P25100 2/20 0.64
OPRM1 known ✓ P35372 2/20 0.64
OPRD1 known ✓ P41143 2/20 0.64
ADRA2C known ✓ P18825 1/20 0.64
MAOA known ✓ P21397 1/20 0.64
MAOB known ✓ P27338 1/20 0.64
LMNA P02545 7/20 1.00
IDO1 P14902 9/20 0.88
CYP2C9 P11712 8/20 0.88
CYP3A4 P08684 8/20 0.88

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Enilconazole SCHEMBL15756772 1.00 LMNA (1.00) LMNAIDO1CYP2C9CYP3A4CYP1A2
Enilconazole SCHEMBL15757117 1.00 LMNA (1.00) LMNAIDO1CYP2C9CYP3A4CYP1A2
Enilconazole SCHEMBL15756834 1.00 LMNA (1.00) LMNAIDO1CYP2C9CYP3A4CYP1A2
Enilconazole SCHEMBL8817070 0.94 IDO1 (1.00) LMNAIDO1CYP2C9CYP3A4CYP1A2
Enilconazole SCHEMBL22498 0.94 IDO1 (1.00) LMNAIDO1CYP2C9CYP3A4CYP1A2
Enilconazole SCHEMBL7913333 0.94 IDO1 (1.00) LMNAIDO1CYP2C9CYP3A4CYP1A2
Enilconazole SCHEMBL29608451 0.94 IDO1 (1.00) LMNAIDO1CYP2C9CYP3A4CYP1A2
Enilconazole SCHEMBL29394655 0.94 IDO1 (1.00) LMNAIDO1CYP2C9CYP3A4CYP1A2
Enilconazole SCHEMBL20472254 0.94 IDO1 (1.00) LMNAIDO1CYP2C9CYP3A4CYP1A2
Enilconazole SCHEMBL28210284 0.93 IDO1 (0.93) LMNAIDO1CYP2C9CYP3A4CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 6296 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026105160-A1 NOVEL AGROCHEMICAL COMPOSITION COMPRISING 3-SUBSTITUTED PHENYLAMIDINE COMPOUNDS AND USE THEREOF PI INDUSTRIES LTD. (IN) 2026-05-21 WO claimed
EP-4114183-B1 FUNGICIDAL COMPOSITIONS SYNGENTA CROP PROTECTION AG (CH) 2026-02-25 EP claimed
EP-3060043-B1 PESTICIDAL COMPOSITIONS AND RELATED METHODS CORTEVA AGRISCIENCE LLC (US) 2025-11-26 EP claimed
EP-4646108-A1 TERNARY COMPOSITION COMPRISING 3-SUBSTITUTED PHENYLAMIDINE COMPOUNDS AND USE THEREOF PI Industries Ltd. (IN) 2025-11-12 EP claimed
EP-4384016-B1 ACTIVE COMPOUND COMBINATIONS AND FUNGICIDE COMPOSITIONS COMPRISING THOSE BAYER AG (DE) 2025-09-03 EP claimed
US-12336537-B2 Fungicidal compositions SYNGENTA CROP PROTECTION AG (CH) 2025-06-24 US claimed
WO-2025098874-A1 ACTIVE COMPOUND COMBINATIONS HAVING FUNGICIDAL/INSECTICIDAL/ACARICIDAL PROPERTIES BAYER AKTIENGESELLSCHAFT (DE) 2025-05-15 WO claimed
US-20250098677-A1 FUNGICIDAL COMPOSITIONS SYNGENTA CROP PROTECTION AG (CH) 2025-03-27 US claimed
CN-115379759-B Method for controlling pests, pest control agent composition, and pest control agent set 日本曹达株式会社 2025-03-14 CN claimed
US-20250040552-A1 FUNGICIDAL COMPOSITIONS SYNGENTA CROP PROTECTION AG (CH) 2025-02-06 US claimed
WO-2006094127-A1 WOOD PRESERVATIVE FORMULATIONS COMPRISING DICHLOROPHEN OSMOSE, INC. (US) 2006-09-08 WO claimed
EP-1424893-B1 FUNGICIDAL MIXTURE CONTAINING ARYLAMIDINE DERIVATIVES BAYER CROPSCIENCE SA (FR) 2006-04-19 EP claimed
US-20040241098-A1 Fungicidal mixture containing arylamidine derivatives BAYER CROPSCIENCE S.A. (FR) 2004-12-02 US claimed
EP-1113727-A1 FOOD COATINGS Janssen Pharmaceutica N.V. (BE) 2001-07-11 EP claimed
WO-2000016644-A1 FOOD COATINGS JANSSEN PHARMACEUTICA N.V. (BE) 2000-03-30 WO claimed
EP-0986965-A1 Antifungal food coatings JANSSEN PHARMACEUTICA N.V. (BE) 2000-03-22 EP claimed
EP-0113254-B1 ANTIMICROBIAL NON-WOVEN FABRIC MICROBAN PRODUCTS COMPANY (US) 1987-10-07 EP claimed
US-4533435-A Antimicrobial paper MICROBAN PRODUCTS COMPANY (US) 1985-08-06 US claimed
EP-0113254-A1 Antimicrobial non-woven fabric MICROBAN PRODUCTS COMPANY (US) 1984-07-11 EP claimed
US-4401712-A Antimicrobial non-woven fabric TULTEX CORPORATION (US) 1983-08-30 US claimed