SCHEMBL4165449

SCHEMBL4165449

CCS(=O)(=O)c1ccccc1-c1cccc(-c2nc3c(C(F)(F)F)cccc3cc2C)c1

nearest known ligand 0.44

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 13/20 0.44
NR1H3 Q13133 12/20 0.44
SCN9A Q15858 3/20 0.38
ALOX5AP P20292 1/20 0.38
FEN1 P39748 1/20 0.38
ATM Q13315 1/20 0.37
PIK3CD O00329 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27786939 0.89 NR1H2 (0.46) NR1H2NR1H3SCN9AATM
SCHEMBL28780848 0.85 NR1H2 (0.39) NR1H2NR1H3ATMPIK3CD
SCHEMBL4165748 0.85 SCN9A (0.46) NR1H2NR1H3SCN9AALOX5APFEN1
SCHEMBL27765402 0.83 NR1H2 (0.40) NR1H2NR1H3ATMPIK3CD
SCHEMBL27765245 0.83 NR1H2 (0.46) NR1H2NR1H3SCN9AALOX5APFEN1
SCHEMBL4165443 0.82 NR1H2 (0.44) NR1H2NR1H3ATMPIK3CD
SCHEMBL4166168 0.82 NR1H2 (0.48) NR1H2NR1H3SCN9A
SCHEMBL28780850 0.80 NR1H2 (0.41) NR1H2NR1H3ATM
SCHEMBL27765403 0.79 NR1H2 (0.40) NR1H2NR1H3
SCHEMBL4174648 0.78 NR1H2 (0.46) NR1H2NR1H3SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101541751-A Quinoline compounds WYETH CORP (US) 2009-09-23 CN claimed
CN-101541751-A Quinoline compounds WYETH CORP (US) 2009-09-23 CN disclosed
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP disclosed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO disclosed