SCHEMBL4166168

SCHEMBL4166168

CCS(=O)(=O)c1ccc(-c2cccc(-c3nc4c(C(F)(F)F)cccc4cc3C)c2)c(Cl)c1

nearest known ligand 0.48

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 12/20 0.48
NR1H3 Q13133 9/20 0.48
RORC P51449 3/20 0.41
PTGDR2 Q9Y5Y4 3/20 0.38
SCN9A Q15858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4162285 0.93 NR1H2 (0.44) NR1H2NR1H3RORC
SCHEMBL4167143 0.90 NR1H2 (0.47) NR1H2NR1H3
SCHEMBL4165449 0.82 NR1H2 (0.44) NR1H2NR1H3SCN9A
SCHEMBL4166161 0.80 NR1H2 (0.46) NR1H2NR1H3RORC
SCHEMBL27765402 0.78 NR1H2 (0.40) NR1H2NR1H3RORC
SCHEMBL27765403 0.76 NR1H2 (0.40) NR1H2NR1H3RORC
SCHEMBL27786939 0.75 NR1H2 (0.46) NR1H2NR1H3SCN9A
SCHEMBL4165443 0.74 NR1H2 (0.44) NR1H2NR1H3RORC
SCHEMBL4162283 0.74 NR1H2 (0.41) NR1H2NR1H3RORC
SCHEMBL28780850 0.72 NR1H2 (0.41) NR1H2NR1H3RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP disclosed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO disclosed