SCHEMBL27765403

SCHEMBL27765403

CCS(=O)(=O)c1ccc(-c2ccccc2)c(Cl)c1-c1nc2c(C(F)(F)F)cccc2cc1C

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 12/20 0.40
NR1H3 Q13133 11/20 0.40
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
DDR1 Q08345 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
RORC P51449 1/20 0.35
ESR1 P03372 1/20 0.35
ENPP1 P22413 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27765096 0.90 NR1H2 (0.41) NR1H2NR1H3ESR1ENPP1
SCHEMBL28780850 0.89 NR1H2 (0.41) NR1H2NR1H3DDR1RORCESR1
SCHEMBL27786978 0.83 KDM4E (0.43) NR1H2NR1H3KDM4EALDH1A1HPGD
SCHEMBL4165443 0.80 NR1H2 (0.44) NR1H2NR1H3CYP1A2CYP3A4CYP2C9
SCHEMBL4166161 0.79 NR1H2 (0.46) NR1H2NR1H3CYP1A2CYP3A4CYP2D6
SCHEMBL4165449 0.79 NR1H2 (0.44) NR1H2NR1H3
SCHEMBL27765402 0.79 NR1H2 (0.40) NR1H2NR1H3KDM4EALDH1A1HPGD
SCHEMBL4166168 0.76 NR1H2 (0.48) NR1H2NR1H3RORC
SCHEMBL4162283 0.75 NR1H2 (0.41) NR1H2NR1H3CYP1A2CYP3A4CYP2D6
SCHEMBL28780848 0.75 NR1H2 (0.39) NR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101541751-A Quinoline compounds WYETH CORP (US) 2009-09-23 CN claimed
CN-101541751-A Quinoline compounds WYETH CORP (US) 2009-09-23 CN disclosed