Mitindomide

Mitindomide

SCHEMBL4171

O=C1NC(=O)[C@H]2[C@H]3C=C[C@@H]([C@@H]12)[C@@H]1[C@H]2C(=O)NC(=O)[C@H]2[C@H]31

nearest known ligand 0.43

Full drug profile on Sugi Atlas →

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.43
SMN1; SMN2 Q16637 2/20 0.35
TSHR P16473 1/20 0.32
CASP1 P29466 1/20 0.32
BRCA1 P38398 1/20 0.32
CASP7 P55210 1/20 0.32
HBB P68871 1/20 0.32
HSD17B10 Q99714 1/20 0.32
GAA P10253 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
MCL1 Q07820 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Mitindomide SCHEMBL19411825 1.00 ALDH1A1 (0.43) ALDH1A1SMN1; SMN2TSHRCASP1BRCA1
SCHEMBL2826555 0.86 ALDH1A1 (0.48) ALDH1A1SMN1; SMN2TSHRCASP1BRCA1
SCHEMBL9526176 0.83 ALDH1A1 (0.46) ALDH1A1TSHRCASP1BRCA1CASP7
SCHEMBL17343101 0.83 ALDH1A1 (0.46) ALDH1A1TSHRCASP1BRCA1CASP7
SCHEMBL9051575 0.75 ALDH1A1 (0.75) ALDH1A1SMN1; SMN2
SCHEMBL9527329 0.75 ALDH1A1 (0.56) ALDH1A1SMN1; SMN2TSHRCASP1BRCA1
SCHEMBL3158529 0.72 POLB (0.40) ALDH1A1TSHRCASP1BRCA1CASP7
SCHEMBL14563304 0.70 ALDH1A1 (0.41) ALDH1A1SMN1; SMN2TSHRCASP1BRCA1
SCHEMBL22260783 0.70 ALDH1A1 (0.45) ALDH1A1SMN1; SMN2TSHRCASP1BRCA1
SCHEMBL20043769 0.70 ALDH1A1 (0.45) ALDH1A1SMN1; SMN2TSHRCASP1BRCA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 9733 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260116861-A1 ISOXAZOLE HYDROXAMIC ACIDS AS HISTONE DEACETYLASE 6 INHIBITORS THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2026-04-30 US claimed
US-12522572-B2 Isoxazole hydroxamic acids as histone deacetylase 6 inhibitors THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2026-01-13 US claimed
EP-4524131-A1 SMALL MOLECULES FOR TREATING CANCER, INHABITING CHEMOKINE ACTIVITY AND/OR INDUCING CELL DEATH AlonBio Ltd. (IL) 2025-03-19 EP claimed
US-12202803-B2 Small molecules for treating cancer, inhibiting chemokine activity and/or inducing cell death ALONBIO LTD. (IL) 2025-01-21 US claimed
US-20240343697-A1 ISOXAZOLE HYDROXAMIC ACIDS AS HISTONE DEACETYLASE 6 INHIBITORS THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2024-10-17 US claimed
US-12109219-B2 Cannabinoid receptor modulators ARENA PHARMACEUTICALS, INC. (US) 2024-10-08 US claimed
WO-2024162488-A1 PHARMACEUTICAL COMPOSITION COMPRISING CUCURBITACIN D FOR PREVENTING OR TREATING NEUROPATHIC PAIN 주식회사 재인알앤피 2024-08-08 WO claimed
EP-4401780-A1 AMORPHOUS PHOTOSENSITIZING PARTICLES, METHODS FOR THE PREPARATION THEREOF, AND METHODS FOR THE USE THEREOF University of Maryland, College Park (US) 2024-07-24 EP claimed
WO-2024026505-A2 DISRUPTION OF TELOCYTE ACTIVITY PATEL AMIT (US) 2024-02-01 WO claimed
US-20240002347-A1 SMALL MOLECULES FOR TREATING CANCER, INHIBITING CHEMOKINE ACTIVITY AND/OR INDUCING CELL DEATH ALONBIO LTD. (IL) 2024-01-04 US claimed
US-20040092583-A1 Treatment for inhibiting neoplastic lesions SHANAHAN-PRENDERGAST ELIZABETH (IE) 2004-05-13 US claimed
EP-1351678-A2 TREATMENT FOR INHIBITING NEOPLASTIC LESIONS USING INCENSOLE AND/OR FURANOGERMACRENS Shanahan-Prendergast, Elizabeth (IE) 2003-10-15 EP claimed
WO-2002053138-A2 TREATMENT FOR INHIBITING NEOPLASTIC LESIONS USING INCENSOLE AND/OR FURANOGERMACRENS SHANAHAN-PRENDERGAST ELISABETH (IE) 2002-07-11 WO claimed
US-5776496-A Ultrasmall porous particles for enhancing ultrasound back scatter UNIVERSITY OF ROCHESTER (US) 1998-07-07 US claimed
EP-0544657-A4 METHOD FOR MAKING UNIFORMLY-SIZED PARTICLES FROM INSOLUBLE COMPOUNDS 1993-08-04 EP claimed
EP-0544657-A1 METHOD FOR MAKING UNIFORMLY-SIZED PARTICLES FROM INSOLUBLE COMPOUNDS THE UNIVERSITY OF ROCHESTER (US) 1993-06-09 EP claimed
WO-1992003380-A1 METHOD FOR MAKING UNIFORMLY-SIZED PARTICLES FROM INSOLUBLE COMPOUNDS THE UNIVERSITY OF ROCHESTER (US) 1992-03-05 WO claimed
EP-0454773-A1 NOVEL PRODRUG DERIVATIVES OF BIOLOGICALLY ACTIVE AGENTS CONTAINING HYDROXYL GROUPS OR NH-ACIDIC GROUPS Bundgaard, Hans (DK) 1991-11-06 EP claimed
US-4997454-A Precipitation THE UNIVERSITY OF ROCHESTER (US) 1991-03-05 US claimed
WO-1990008128-A1 NOVEL PRODRUG DERIVATIVES OF BIOLOGICALLY ACTIVE AGENTS CONTAINING HYDROXYL GROUPS OR NH-ACIDIC GROUPS BUNDGAARD HANS (DK) 1990-07-26 WO claimed