SCHEMBL4175965

SCHEMBL4175965

COc1ccccc1C#Cc1cc(C(N)=O)c(OC(C)C)c(C(CO)Cc2c[nH]c3ccncc23)c1.NC(CO)Cc1c[nH]c2cccnc12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 19/20 0.36
SCN9A Q15858 1/20 0.31
EEF2K O00418 1/20 0.31
DYRK3 O43781 1/20 0.31
PRKD3 O94806 1/20 0.31
CSNK1D P48730 1/20 0.31
CLK2 P49760 1/20 0.31
GSK3A P49840 1/20 0.31
RPS6KA3 P51812 1/20 0.31
PRKCD Q05655 1/20 0.31
STK3 Q13188 1/20 0.31
CAMK2B Q13554 1/20 0.31
CAMK2G Q13555 1/20 0.31
DYRK1A Q13627 1/20 0.31
ERBB4 Q15303 1/20 0.31
PRKD2 Q9BZL6 1/20 0.31
CLK4 Q9HAZ1 1/20 0.31
PIM2 Q9P1W9 1/20 0.31
AKT3 Q9Y243 1/20 0.31
PDPK1 O15530 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Tryptophanol SCHEMBL4785476 0.75 AKT1 (0.42) AKT1SCN9AEEF2KDYRK3PRKD3
SCHEMBL3943487 0.71 ROCK2 (0.38)
SCHEMBL13911141 0.71 ROCK2 (0.38) AKT1
SCHEMBL3941491 0.71 ROCK2 (0.38) AKT1
SCHEMBL4785471 0.67 ITGB2 (0.44)
SCHEMBL3944155 0.66 ROCK2 (0.38)
SCHEMBL13911177 0.66 ROCK2 (0.38)
SCHEMBL3939139 0.65 ITGB2 (0.41)
SCHEMBL4632690 0.64 HDAC3 (0.44)
SCHEMBL4633717 0.64 HDAC3 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009013354-A1 ARYLMETHYLENE SUBSTITUTED N-ACYL-β-AMINO ALCOHOLS BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2009-01-29 WO claimed